Synthesis and bioactivity evaluation of rhodanine derivatives as potential anti-bacterial agents
European Journal of Medicinal Chemistry, 2012Five series of (Z)-5-(4-(2-oxo-2-phenylethoxy)benzylidene)-2-thioxothiazolidin-4-one derivatives (I-V) were synthesized, characterized, and evaluated for their anti-bacterial activity. Most of the synthesized compounds showed potent inhibition against several Gram-positive bacteria (including multidrug-resistant clinical isolates) with MIC values in ...
Ming-Xia, Song +7 more
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Quinolone‐Rhodanine Hybrid Compounds: Synthesis and Biological Evaluation as Anti‐Bacterial Agents
ChemistrySelect, 2022Abstract As potential antimicrobial agents, 4‐fluoroaniline and diethyl (ethoxymethylene)malonate were used to efficiently synthesize a new quinolone (3‐9) series. The 1 HNMR and 13 C NMR, IR ...
Yıldız Uygun Cebeci +1 more
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Therapeutic Potential of Alkaloids as Anti-Bacterial Agents: Drugs of Future
Current Bioactive Compounds, 2019Bacterial infections remain a major threat to the world community in terms of both morbidity and mortality. Indeed, bacterial infections are accountable for millions of fatalities around the globe. Additionally, these bacterial infections represent a notable burden, in particular, for children living in less-developed regions of the world.
Aini Pervaiz, Haroon Khan, Surriya Amin
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Synthesis and biological evaluation of resveratrol analogues as anti-bacterial agents
2011 IEEE International Symposium on IT in Medicine and Education, 2011Resveratrol (3,5,4′-trihydroxy-trans-stilbene) is a stilbenoid, a type of natural phenol, and a phytoalexin produced naturally by several kinds of plants when under attack by pathogens such as bacteria or fungi which exerts a variety of biological activities.
null Rui Cao +5 more
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ChemInform Abstract: SYNTHESIS OF 10‐THIOAMINOPTERIN, A POTENT ANTI‐BACTERIAL AGENT
Chemischer Informationsdienst, 1975AbstractAus dem Phthalimid (I) und dem p‐Carbomethoxy‐thiophenol (II) werden die Oxime ‐ (IIIa) und (IIIb) hergestellt.
M. G. NAIR +3 more
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The use of FTIR microscopy for the evaluation of anti-bacterial agents activity
Journal of Photochemistry and Photobiology B: Biology, 2009FTIR spectroscopy has been used by chemists as a powerful tool to characterize inorganic and organic compounds. In this study we examined the potential of FTIR microspectroscopy for early evaluation of the efficiency of anti-bacterial therapy. For this purpose, the effect of caffeic acid phenethyl ester (CAPE) and ampicillin on the development of ...
Mahmoud, Huleihel +2 more
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Boc‐Protected Phenylalanine and Tryptophan‐Based Dipeptides: A Broad Spectrum Anti‐Bacterial Agent
BiopolymersABSTRACTDipeptides were constructed using hydrophobic amino acid residues following AMP prediction. After that Boc‐modification was performed on the screened peptides and finally Boc‐Phe‐Trp‐OMe and Boc‐Trp‐Trp‐OMe were synthesized. Even though no inhibition zones were observed in agar well diffusion assays, minimum inhibitory concentration (MIC ...
Arpita Halder +4 more
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Molecular imaging in oncology: Current impact and future directions
Ca-A Cancer Journal for Clinicians, 2022Steven P Rowe, Martin G Pomper
exaly
Synthesis of 10-thioaminopterin: A potent anti-bacterial agent
Tetrahedron Letters, 1975M.G. Nair +3 more
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