Results 191 to 200 of about 20,936 (236)

Insights into the Design of MYC-Targeting Proteolysis Targeting Chimeras (PROTACs). [PDF]

open access: yesMolecules
Alfayomy AM   +6 more
europepmc   +1 more source

Indole Peptidomimetics Show Potent and Selective Activity against Drug-Resistant <i>Plasmodium falciparum</i>. [PDF]

open access: yesACS Omega
Januário MAP   +8 more
europepmc   +1 more source

Intercalation of Benzamide into Kaolinite

Journal of Colloid and Interface Science, 2000
Well-crystallized kaolinite (K) was initially reacted at 60 degrees C with a water/dimethylsulfoxide (DMSO) mixture and the resulting intercalation derivative (K-DMSO) was characterized by powder X-ray diffractometry (PXRD), thermal analysis (simultaneous TG and DSC), and Fourier-transformed infrared spectroscopy (FTIR).
Luiz Pereira Ramos, Fernando Wypych
exaly   +3 more sources

Synthesis of benzamide derivatives and their evaluation as antiprion agents

open access: yesBioorganic and Medicinal Chemistry, 2012
A new set of 5-(2-(pyrrolidin-1-yl)acetamido)-N-butyl-2-(substituted)benzamide and 5-(2-(piperidin-1-yl)acetamido)-N-butyl-2-(substituted) benzamide derivatives were synthesized in which as structural features the 2-(1-pyrrolidinyl)- or 2-(1-piperidyl ...
Martin Eiden   +2 more
exaly   +2 more sources

Mechanochemically Induced Conversion of Crystalline Benzamide Polymorphs by Seeding

open access: yesAngewandte Chemie - International Edition, 2016
Benzamide has been known for its polymorphism for almost 200 years.Three polymorphic forms are described. To date,itwas only possible to crystallizeametastable form in amixture together with the thermodynamically most stable form I.
Klaus Rademann, Franziska Emmerling
exaly   +2 more sources

Pharmacological Classification of Benzamides

Acta Psychiatrica Scandinavica, 1984
Abstract The problem of classifying benzamides is, in general, the same as classifying neuroleptics. A pharmacological classification of neuroleptics can be established on the basis of the following criteria‐ specificity of action on dopaminergic receptors‐ penetration into the CNS‐ dopaminergic profile in the CNS• relative binding with respect to ...
A J, Puech, Y, Lecrubier, P, Simon
openaire   +2 more sources

ortho-Arylation of Benzamides

Organic Letters, 2006
[reaction: see text] A simple method for the direct ortho-arylation of benzoic acid amides has been developed. The palladium-catalyzed reactions proceed in trifluoroacetic acid and require the presence of stoichiometric silver acetate. This presents an alternative to the currently used ortho-lithiation strategies for the synthesis of arylated benzoic ...
Dmitry, Shabashov, Olafs, Daugulis
openaire   +2 more sources

Alkylating benzamides with melanoma cytotoxicity

Melanoma Research, 2004
Radioiodinated N-(2-(diethylamino)ethyl)benzamides have recently been discovered as selective agents for melanotic melanoma and are used for scintigraphic imaging in nuclear medicine. Owing to the high binding capacity, benzamide derivatives conjugated with alkylating cytostatics were synthesized and tested for their potential for targeted drug ...
Markus, Wolf   +6 more
openaire   +2 more sources

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