Results 91 to 100 of about 5,260 (223)
Melanin-concentrating hormone receptor 1 antagonists: Synthesis, structure–activity relationship, docking studies, and biological evaluation of 2,3,4,5-tetrahydro-1H-3-benzazepine derivatives
, 2011 Shizuo Kasai, Masahiro Kamaura, Makoto Kamata, Kazuyoshi Aso, Hitomi Ogino, Yoshihide Nakano, Kaoru Watanabe, Tomoko Kaisho, Michiko Tawada, Yasutaka Nagisa, Shiro Takekawa, Koki Kato, Nobuhiro Suzuki, Yuji Ishihara +13 moreopenalex +1 more sourceThe discovery and optimisation of benzazepine sulfonamide and sulfones as potent agonists of the motilin receptor
, 2009 James M. Bailey, J. Scott, Jonathan B. Basilla, Victoria J. Bolton, Izzy Boyfield, David G. Evans, Étienne Fleury, Tom D. Heightman, Emma M. Jarvie, Kirk Lawless, Kim L. Matthews, Fiona C. McKay, Hindy Mok, Alison I. Muir, Barry S. Orlek, Gareth J. Sanger, Geoffrey Stemp, Alexander J. Stevens, Mervyn Thompson, John M. Ward, Kalindi Vaidya, Susan M. Westaway +21 moreopenalex +1 more sourceFragment-Based Screening Identifies New Quinazolinone-Based Inositol Hexakisphosphate Kinase (IP6K) Inhibitors. [PDF]
ACS Med Chem Lett, 2023 Heitmann T, Liao G, de León P, Ernst G, Buchler I, Wei H, Shlevkov E, Brown D, Fitzek M, Collier M, Smith DM, Barrow JC. +11 moreeuropepmc +1 more sourceIdentification of clinical candidates from the benzazepine class of histamine H3 receptor antagonists
, 2013 David M. Wilson, James Apps, Nicholas Bailey, Mark J. Bamford, I.J.M. Beresford, Kim Brackenborough, Michael A. Briggs, Stephen Brough, Andrew R. Calver, Barry Crook, Rebecca K. Davis, Robert P. Davis, Susannah Davis, David K. Dean, Leanne Harris, Teresa Heslop, Vicky Holland, Philip D. Jeffrey, Terrance A. Panchal, Christopher A. Parr, Nigel Quashie, Joanne Schogger, Sanjeet S. Sehmi, Tania O. Stean, Jon G.A. Steadman, Brenda Trail, Jeffrey Wald, Angela Worby, Andrew K. Takle, Jason Witherington, Andrew D. Medhurst +30 moreopenalex +1 more source