Photoinduced Copper‐Catalyzed Cross‐Coupling of Acylsilanes with Heteroarenes via Bimetallic Relay [PDF]
Advanced ScienceThe transition metal‐catalyzed direct coupling reactions involving electron‐rich Fischer carbene species are largely underdeveloped and remain a big challenge.
Long Zheng +3 more
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A Mechanism Study on the (+)-ESI-TOF/HRMS Fragmentation of Some PPI Prazoles and Their Related Substances [PDF]
Molecules, 2023 Fragmentation mechanisms of some prazoles and their related substances were newly investigated in this paper via positive mode ESI-TOF HRMS1 and HRMS2. Some novel fragmentation rules or ions were found or detected in the research.
Luhong Wang +4 more
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Anti-Tumoral Effects of a (1H-Pyrrol-1-yl)Methyl-1H-Benzoimidazole Carbamate Ester Derivative on Head and Neck Squamous Carcinoma Cell Lines [PDF]
Pharmaceuticals, 2021 Nocodazole is an antineoplastic agent that exerts its effects by depolymerizing microtubules. Herein we report a structural analog of nocodazole, a (1H-pyrrol-1-yl)methyl-1H-benzoimidazole carbamate ester derivative, named RDS 60.
Alice Nicolai +14 more
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Towards discovery of new leishmanicidal scaffolds able to inhibit Leishmania GSK-3 [PDF]
Journal of Enzyme Inhibition and Medicinal Chemistry, 2020 Previous reports have validated the glycogen synthase kinase-3 (GSK-3) as a druggable target against the human protozoan parasite Leishmania. This prompted us to search for new leishmanicidal scaffolds as inhibitors of this enzyme from our in-house ...
Paula Martínez de Iturrate +9 more
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N-Benzoimidazole/Oxadiazole Hybrid Universal Electron Acceptors for Highly Efficient Exciplex-Type Thermally Activated Delayed Fluorescence OLEDs [PDF]
Frontiers in Chemistry, 2019 Recently, donor/acceptor type exciplex have attracted considerable interests due to the low driving voltages and small singlet-triplet bandgaps for efficient reverse intersystem crossing to achieve 100% excitons for high efficiency thermally activated ...
Wenbo Yuan +5 more
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Beilstein Journal of Organic Chemistry, 2023 1,3-Dimethyl-2,3-dihydrobenzo[d]imidazoles, 1H, and 1,1',3,3'-tetramethyl-2,2',3,3'-tetrahydro-2,2'-bibenzo[d]imidazoles, 12, are of interest as n-dopants for organic electron-transport materials.
Swagat K. Mohapatra +8 more
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Synthesis and anticancer properties of 5-(1H-benzoimidazol-2-ylmethylene)-4-oxo-2-thioxothiazolidin-3-ylcarboxilic acids [PDF]
Pharmacia, 2021 The reaction of 1H-benzoimidazole-2-carbaldehyde with 4-oxo-2-thioxothiazolidin-3-ylcarboxilic acids was studied and the combinatorial library of 5-(1H-benzoimidazol-2-ylmethylene)-4-oxo-2-thioxothiazolidin-3-ylcarboxilic acids has been prepared.
Volodymyr Horishny +2 more
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Catalysis Communications, 2021 An efficient I2/TBHP promoted isocyanide insertion cyclization reaction for the synthesis of quinazolines-fused benzoimidazole was reported. The synthesized compounds have a unique potential to use as a selective solvatochromic fluorescence probe for ...
Fereshteh Ahmadi +4 more
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Ethyl 1-(4-fluorobenzyl)-2-(4-methoxyphenyl)-1H-benzo[d]imidazole-5-carboxylate
IUCrData, 2016 The title benzoimidazole derivative, C24H21FN2O3, is T-shaped, with the methoxyphenyl and fluorobenzyl rings inclined to the benzoimidazole ring system by 40.91 (8) and 86.04 (8)°, respectively, indicating that the fluorobenzyl ring system is nearly ...
S. Naveen +5 more
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Acta Crystallographica Section E: Crystallographic Communications, 2017 The side product of the cyclocondensation reaction between ethyl benzimidazole-2-carboxylate and the nitrile imine of the corresponding hydrazonyl chloride, C20H11BrClN5O, crystallized in two crystal forms. Form (1) is a co-crystal of the target compound
Kanan Wahedy +6 more
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