Borylcyclopropanes: Synthetic Strategies and Applications
Angewandte Chemie, EarlyView.Borylcyclopropanes (cyclopropanes bearing a boron substituent) sit at the intersection of two privileged frameworks in synthesis. This review provides the first exhaustive survey of their chemistry, spanning metal–carbene, nucleophilic cyclization, radical, hydroboration, and C─H activation routes, and documenting applications in medicinal chemistry ...
Aiza A. Butt, Joseph M. Ready
wiley +2 more sources
Enhanced "Green Nudging": Tapping the channels of cultural transmission. [PDF]
PLoS OneCordes C, Henkel J.
europepmc +1 more source
Australian Journal of Social Issues, EarlyView.ABSTRACT Nations manufacture non‐belonging of temporary migrants through policy frameworks that produce exclusion. This precarity maximises the economic benefit of temporary migrant labour by minimising their political, social and legal rights. In this paper, we examine how non‐belonging targeting Working Holiday Makers (WHMs) is manufactured in ...
Donna James, Alanna Kamp
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Multicomponent Stapling of Glucagon‐Like Peptide‐1 Enables Receptor‐Guided PROTAC Delivery
Angewandte Chemie, EarlyView.We report a stapled glucagon‐like peptide‐1 (GLP‐1) analogue created via multicomponent tryptophan‐mediated Petasis reaction (TMPR). This strategy yields a stabilised peptide with superior helicity and improved potency. Conjugation to a bromodomain‐containing protein 4 (BRD4) degrader creates the first GLP‐1‐guided targeted protein degrader (PROTAC ...
Jan L. Venne +5 more
wiley +2 more sources
The Application of Wargaming in the Nuclear Emergency Preparedness Phase to Improve Urgent and Early Phase Response Planning and Decision Making. [PDF]
Health PhysBuchanan K, Bergman L, Nsengiyumva D.
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Air Pollution, Body Composition, and Vascular Age in Southern Switzerland: A Cross-Sectional Population Study. [PDF]
J Clin MedPasini M +6 more
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Values of Stakeholders Involved in Applying Surveillance Technology for People With Dementia in Nursing Homes: Scoping Review. [PDF]
JMIR Agingvan Gaans-Riteco D, Stoop A, Wouters E.
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Gender and residential differences in sleep quality among Chinese adolescents aged 13-18 years. [PDF]
PLoS OneKang X, Li J, Wu H.
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Health Risk Assessment of Residents' Exposure to Air Pollutants around the Sinpyeong-Jangrim Industrial Complex in Busan. [PDF]
ToxicsJung JY +5 more
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GIS-based soil bearing capacity zonation maps for the Dhaka metropolitan development plan (DMDP) area, Bangladesh. [PDF]
Sci RepRahman MS, Alajlan ZS, Ansary MA.
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