Results 221 to 230 of about 125,338 (250)

Insights into MAPK p38α DFG flip mechanism by accelerated molecular dynamics

Bioorganic and Medicinal Chemistry, 2010
Francesca De Rienzo, M Cristina Menziani   +1 more
exaly  

Enhanced selectivity profile of pyrazole-urea based DFG-out p38α inhibitors

Bioorganic and Medicinal Chemistry Letters, 2010
Haile Tecle, Jessie M English
exaly  

Preparation of activated flavor precursor DFG, N-(1-deoxy-1-fructosylglycine) by combination of vacuum evaporation and closed system heating steps

Food Chemistry, 2018
Tomáš Davídek, Karin Kraehenbuehl
exaly  

The dynamic switch mechanism that leads to activation of LRRK2 is embedded in the DFGψ motif in the kinase domain

Proceedings of the National Academy of Sciences of the United States of America, 2019
Friedrich W Herberg, Sven H Schmidt, Matthias Joseph Knape   +2 more
exaly  

DFG-in and DFG-out homology models of TrkB kinase receptor: Induced-fit and ensemble docking

Journal of Molecular Graphics and Modelling, 2010
Pierfausto Seneci, Anna Bernardi, Črtomir Podlipnik   +2 more
exaly  

An SFG/DFG investigation of CN− adsorption at an Au electrode in 1-butyl-1-methyl-pyrrolidinium bis(trifluoromethylsulfonyl) amide ionic liquid

Electrochemistry Communications, 2010
Adriana Ispas, Christophe Humbert, Andreas Bund   +2 more
exaly  

Discovery of a Type III Inhibitor of LIM Kinase 2 That Binds in a DFG-Out Conformation

ACS Medicinal Chemistry Letters, 2015
Nicole Goodwin, Giovanni Cianchetta, Jason Allen   +2 more
exaly  

Sorafenib inhibits p38α activity in colorectal cancer cells and synergizes with the DFG-in inhibitor SB202190 to increase apoptotic response

Cancer Biology and Therapy, 2012
Anna Napoli, Alberto Del Rio, Cristiano Simone   +2 more
exaly  

Identification and Characterization of Small‐Molecule Inhibitors to Selectively Target the DFG‐in over the DFG‐out Conformation of the B‐Raf Kinase V600E Mutant in Colorectal Cancer

Archiv Der Pharmazie, 2016
Jinshui Zhu
exaly  

Azaindole-Based Inhibitors of Cdc7 Kinase: Impact of the Pre-DFG Residue, Val 195

ACS Medicinal Chemistry Letters, 2013
Kent Stewart, John E Harlan
exaly