Results 171 to 180 of about 13,967 (254)

Rational Design, Synthesis and Pharmacological Evaluation of Chalcones as Dual-Acting Compounds-Histamine H₃ Receptor Ligands and MAO-B Inhibitors. [PDF]

Int J Mol Sci
Łażewska D, Doroz-Płonka A, Kuder K, Siwek A, Wagner W, Karnafał-Ziembla J, Olejarz-Maciej A, Wolak M, Głuch-Lutwin M, Mordyl B, Osiecka O, Juszczak M, Woźniak K, Więcek M, Latacz G, Stasiak A.   +15 more
europepmc   +1 more source

Identification of clinical candidates from the benzazepine class of histamine H3 receptor antagonists

, 2013
David M. Wilson, James Apps, Nicholas Bailey, Mark J. Bamford, I.J.M. Beresford, Kim Brackenborough, Michael A. Briggs, Stephen Brough, Andrew R. Calver, Barry Crook, Rebecca K. Davis, Robert P. Davis, Susannah Davis, David K. Dean, Leanne Harris, Teresa Heslop, Vicky Holland, Philip D. Jeffrey, Terrance A. Panchal, Christopher A. Parr, Nigel Quashie, Joanne Schogger, Sanjeet S. Sehmi, Tania O. Stean, Jon G.A. Steadman, Brenda Trail, Jeffrey Wald, Angela Worby, Andrew K. Takle, Jason Witherington, Andrew D. Medhurst   +30 more
openalex   +1 more source

Alleviation of Autophagic Deficits and Neuroinflammation by Histamine H3 Receptor Antagonist E159 Ameliorates Autism-Related Behaviors in BTBR Mice. [PDF]

Pharmaceuticals (Basel)
Thomas SD, Jayaprakash P, Marwan NZHJ, Aziz EABA, Kuder K, Łażewska D, Kieć-Kononowicz K, Sadek B.   +7 more
europepmc   +1 more source

Cloning of Rat Histamine H3 Receptor Reveals Distinct Species Pharmacological Profiles

, 2000
Timothy W. Lovenberg, Jayashree Pyati, Hong Chang, Sandy J. Wilson, Mark G. Erlander   +4 more
openalex   +1 more source

Reproductive and fetal toxicity studies of histamine H3 receptor antagonist DL76 used in mice to prevent maximal electroshock-induced seizure. [PDF]

Front Pharmacol
Bastaki SM, Abdulrazzaq YM, Zidan MA, Shafiullah M, Alaryani SG, Alnuaimi FA, Adeghate E, Mohsin S, Akour A, Siwek A, Łażewska D, Kieć-Kononowicz K, Sadek B.   +12 more
europepmc   +1 more source

Histamine H₃ Receptor Isoforms: Insights from Alternative Splicing to Functional Complexity. [PDF]

Biomolecules
Gao M, Ooms JF, Leurs R, Vischer HF.
europepmc   +1 more source

Histamine H3 Receptor Promotes Cell Survival via Regulating PKA/CREB/CDKN1A Signal Pathway in Hepatocellular Carcinoma. [PDF]

Onco Targets Ther, 2020
Zhang C, Yu Y, Ma L, Fu P.
europepmc   +1 more source

Trans-4-methyl-3-imidazoyl pyrrolidine as a potent, highly selective histamine H3 receptor agonist in vivo

, 1998
Neng‐Yang Shih, Robert Aslanian, Andrew T. Lupo, Steve Orlando, John J. Piwinski, Michael J. Green, Ashit K. Ganguly, Robert West, S. Tozzi, William Kreutner, John A. Hey   +10 more
openalex   +1 more source

A new class of histamine H3-Receptor antagonists: synthesis and structure–Activity relationships of 7,8,9,10-Tetrahydro-6H-cyclohepta[b]quinolines

, 2003
Sean Turner, Timothy A. Esbenshade, Youssef L. Bennani, Arthur A. Hancock   +3 more
openalex   +1 more source

Effects of thioperamide, an antagonist of histamine H3-receptor, on monoamine levels and monoamine oxidase activity in rat brain.

, 1993
Eiichi Sakurai, Eiko Sakurai, Kazutaka Maeyama, Takehiko Watanabe, Lars Oreland   +4 more
openalex   +1 more source