Results 181 to 190 of about 13,967 (254)

Exploring occupancy of the histamine H₃ receptor by pitolisant in humans using PET. [PDF]

Br J Pharmacol, 2020
Rusjan P, Sabioni P, Di Ciano P, Mansouri E, Boileau I, Laveillé A, Capet M, Duvauchelle T, Schwartz JC, Robert P, Le Foll B.   +10 more
europepmc   +1 more source

The Novel Pimavanserin Derivative ST-2300 with Histamine H₃ Receptor Affinity Shows Reduced 5-HT_2A Binding, but Maintains Antidepressant- and Anxiolytic-like Properties in Mice. [PDF]

Biomolecules, 2022
Venkatachalam K, Zhong S, Dubiel M, Satała G, Sadek B, Stark H.   +5 more
europepmc   +1 more source

Developmentand Preclinical Characterization of [¹⁸F]H3-2406 and [¹⁸F]H3-2407 for Positron EmissionTomography Imaging of the Histamine Subtype‑3 Receptor

Zhendong Song (9731871), Yinlong Li (1884139), Kenneth Dahl (4782936), Zhenkun Sun (1286034), Jiahui Chen (1818361), Xin Zhou (54275), Yabiao Gao (9991754), Jian Rong (598108), Chunyu Zhao (1977382), Katherine Yuan (21725559), Ahmad F. Chaudhary (19923541), Jimmy S. Patel (4453471), Thomas L. Collier (3637486), Chongzhao Ran (222663), Kim S. Muehlfenzl (21725562), Achi Haider (20428250), Charles S. Elmore (2004724), Magnus Schou (1408873), Steven H. Liang (1341546)   +18 more
openalex   +1 more source

AR71, Histamine H₃ Receptor Ligand-In Vitro and In Vivo Evaluation (Anti-Inflammatory Activity, Metabolic Stability, Toxicity, and Analgesic Action). [PDF]

Int J Mol Sci
Stasiak A, Honkisz-Orzechowska E, Gajda Z, Wagner W, Popiołek-Barczyk K, Kuder KJ, Latacz G, Juszczak M, Woźniak K, Karcz T, Szczepańska K, Jóźwiak-Bębenista M, Kieć-Kononowicz K, Łażewska D.   +13 more
europepmc   +1 more source

Covalent Inhibition of the Histamine H₃ Receptor. [PDF]

Molecules, 2019
Wágner G, Mocking TAM, Kooistra AJ, Slynko I, Ábrányi-Balogh P, Keserű GM, Wijtmans M, Vischer HF, de Esch IJP, Leurs R.   +9 more
europepmc   +1 more source

The Neuroprotective Effects of Histamine H3 Receptor Antagonist E177 on Pilocarpine-Induced Status Epilepticus in Rats. [PDF]

Molecules, 2019
Alachkar A, Azimullah S, Ojha SK, Beiram R, Łażewska D, Kieć-Kononowicz K, Sadek B.   +6 more
europepmc   +1 more source

Nasal hyperreactivity and inflammation in perennial allergic rhinitis [PDF]

, 1995
Garrelds, I.M. (Ingrid), Veld, C. (Catharina) in 't   +1 more
core  

The histamine H₃ receptor inverse agonist SAR-152954 reverses deficits in long-term potentiation associated with moderate prenatal alcohol exposure. [PDF]

Alcohol
Goncalves-Garcia M, Davies S, Savage DD, Hamilton DA.   +3 more
europepmc   +1 more source

Histamine H3 Receptor Antagonist Enhances Neurogenesis and Improves Chronic Cerebral Hypoperfusion-Induced Cognitive Impairments. [PDF]

Front Pharmacol, 2019
Wang N, Ma J, Liu J, Wang J, Liu C, Wang H, Liu Y, Yan H, Jiang S.   +8 more
europepmc   +1 more source

Development of a Conformational Histamine H₃ Receptor Biosensor for the Synchronous Screening of Agonists and Inverse Agonists. [PDF]

ACS Sens, 2020
Schihada H, Ma X, Zabel U, Vischer HF, Schulte G, Leurs R, Pockes S, Lohse MJ.   +7 more
europepmc   +1 more source