Results 121 to 130 of about 10,224 (203)

Simultaneous Blockade of Histamine H₃ Receptors and Inhibition of Acetylcholine Esterase Alleviate Autistic-Like Behaviors in BTBR T+ tf/J Mouse Model of Autism. [PDF]

Biomolecules, 2020
Eissa N, Jayaprakash P, Stark H, Łażewska D, Kieć-Kononowicz K, Sadek B.   +5 more
europepmc   +1 more source

Drug-likeness approach of 2-aminopyrimidines as histamine H3 receptor ligands

Drug Design, Development and Therapy, 2014
Bassem Sadek,1 Annemarie Schreeb,2 Johannes Stephan Schwed,2,3 Lilia Weizel,2 Holger Stark3 1Department of Pharmacology and Therapeutics, College of Medicine and Health Sciences, United Arab Emirates University, Al Ain, United Arab Emirates; 2Biocenter ...
Sadek B, Schreeb A, Schwed JS, Weizel L, Stark H   +4 more
doaj  

Simultaneous inhibition of cholinesterase and antagonism of histamine H3 receptors alleviates cognitive deficits and mitigates apoptosis in scopolamine-induced amnesia in mice. [PDF]

Front Behav Neurosci
Ebdah W, Thomas SD, Eissa N, Jayaprakash P, Łażewska D, Kieć-Kononowicz K, Sadek B.   +6 more
europepmc   +1 more source

Development of TASP0410457 (TASP457), a novel dihydroquinolinone derivative as a PET radioligand for central histamine H3 receptors. [PDF]

EJNMMI Res, 2016
Koga K, Maeda J, Tokunaga M, Hanyu M, Kawamura K, Ohmichi M, Nakamura T, Nagai Y, Seki C, Kimura Y, Minamimoto T, Zhang MR, Fukumura T, Suhara T, Higuchi M.   +14 more
europepmc   +1 more source

4-Oxypiperidine Ethers as Multiple Targeting Ligands at Histamine H₃ Receptors and Cholinesterases. [PDF]

ACS Chem Neurosci
Michalska B, Dzięgielewski M, Godyń J, Werner T, Bajda M, Karcz T, Szczepańska K, Stark H, Więckowska A, Walczyński K, Staszewski M.   +10 more
europepmc   +1 more source

The Impact of H1-H4 Receptor Antagonists on the Levels of Selected Oxidative Stress Markers in Liver and Muscle Tissue in an Animal Model of Colitis. [PDF]

Pharmaceuticals (Basel)
Bogielski B, Michalczyk K, Gębski W, Rozpędek K, Szulińska E, Tempka B, Zorychta A, Chełmecka E, Kaczmar E, Głodek P, John J, Nikiel K, Skrzep-Poloczek B, Jochem J, Kieć-Kononowicz K, Łażewska D, Stygar D.   +16 more
europepmc   +1 more source

Activity-restoring mutations in the histamine H₃ receptor increase constitutive activity and reduce structural stability. [PDF]

Protein Sci
Nakajima A, Kaneko H, Oyama K, Kuchiji M, Itakura A, Arai C, Shiroishi M.   +6 more
europepmc   +1 more source

Antihistamines: Beyond just allergy treatment

Vietnam Journal of Science, Technology and Engineering
Histamine and its receptors (H1R-H4R) are involved in several significant physiological processes and pathogenic conditions. Antihistamines, widely recognised as drugs for treating allergies, belong to the H1 antihistamine group, which targets H1R on ...
Hue T. H. Bui, Xuan-Hung Nguyen
doaj  

Letter to the Editor in Response to "Efficacy and Safety of Histamine H3 Receptor Antagonist/Inverse Agonist Including Betahistine for Schizophrenia: A Systematic Review and Meta-Analysis" by Nishii et al. [PDF]

Neuropsychopharmacol Rep
Farhan M.
europepmc   +1 more source

Novel Thiazolobenzodiazepines As Inhibitors of Histamine H3 Receptor [PDF]

ACS Medicinal Chemistry Letters, 2013
openaire   +2 more sources