1,2,3,6-Tetrahydropyridine-4-carboxylic acid (isoguvacine) and related 2-and/or 6-methylated analogues (1-4) were synthesized using the methoxycarbonylation [Pd(OAc)(2), PPh(3), CO, MeOH)] of their corresponding vinylic triflates.
Garrido, F. +5 more
core +1 more source
A concise synthesis and the antibacterial activity of 5,6-dimethoxynaphthalene-2-carboxylic acid
5,6-Dimethoxynaphthalene-2-carboxylic acid was synthesized in 7 steps and with an overall yield of 46%. Bromination of 2-naphthol, and methylation with dimethyl sulfate followed by Friedel-Crafts acylation with AcCl gave 2-acetyl-5-bromo-6 ...
UGUZ, METİN TANSU +3 more
core
A Micronized Crystalline form-R of 2-(3,5-dichloro phenyl) -1,3-benzoxazole-6- carboxylic acid [PDF]
The present invention provides Micronized Crystalline form-R of 2-(3,5- dichloro phenyl)-1,3-benzoxazole-6-carboxylic acid of formula (I) and process for preparation ...
, MSN Laboratories Private Limited, R&D Center; Srinivasan Thirumalai Rajan, Sagyam Rajeshwar Reddy, Kammari Balraju
core +1 more source
The K atom in the title complex, [K(C(10)H(6)NO(2))(C(10)H(7)NO(2))(3)], lies on a twofold rotation axis that relates one N,O-chelating quinoline-2-carboxylic acid to the other; their N and O atoms are cis to each other in the distorted octahedral ...
Ng, S.W.
core +1 more source
Trifluoromethylation of pyridines through skeletal rearrangement. [PDF]
Wang H, Bhaduri N, Greaney MF.
europepmc +1 more source
Tunable Osmium Complexes as pH-Insensitive Redox Reporters for Electrochemical Biosensing. [PDF]
Montón Vicente A +7 more
europepmc +1 more source
Initiating Photocontrolled Atom Transfer Radical Polymerization from a Redox-Activated Functional Group. [PDF]
McClements IF, Driscoll ME, Fors BP.
europepmc +1 more source
Hyperpolarization of Pyridine <sup>15</sup>N-Oxide Molecular Probes Enabled by Parahydrogen. [PDF]
Mei R +8 more
europepmc +1 more source
Programmable regiodivergent light-driven cyclization of acyclic 1,5-dienes unlocks rigid bicyclic architectures. [PDF]
Zhang ZX +6 more
europepmc +1 more source
Novel process for the preparation of 6-hydroxy-2-methylbenzofuran-3-carboxylic acid [PDF]
The present disclosure relates to a novel process for the preparation of 6-hydroxy-2-methylbenzofuran-3-carboxylic acid of formula-2 which is a key intermediate used in the preparation of Fruquintinib.
, MSN Laboratories Private Limited, R&D Center; Hyderabad, India; Srinivasan Thirumalai Rajan; Gade Srinivas Reddy & Surigilla Venkateshwarlu
core

