Results 1 to 10 of about 398,732 (120)

New Deoxycholic Acid Derived Tyrosyl-DNA Phosphodiesterase 1 Inhibitors Also Inhibit Tyrosyl-DNA Phosphodiesterase 2

Molecules, 2021
A series of deoxycholic acid (DCA) amides containing benzyl ether groups on the steroid core were tested against the tyrosyl-DNA phosphodiesterase 1 (TDP1) and 2 (TDP2) enzymes.
Oksana V. Salomatina, Nadezhda S. Dyrkheeva, Irina I. Popadyuk, Alexandra L. Zakharenko, Ekaterina S. Ilina, Nina I. Komarova, Jóhannes Reynisson, Nariman F. Salakhutdinov, Olga I. Lavrik, Konstantin P. Volcho   +9 more
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Design, Synthesis, and Bioactivities of Novel Trifluoromethyl Pyrimidine Derivatives Bearing an Amide Moiety

Frontiers in Chemistry, 2022
Twenty-three novel trifluoromethyl pyrimidine derivatives containing an amide moiety were designed and synthesized through four-step reactions and evaluated for their antifungal, insecticidal, and anticancer properties.
Wenjun Lan, Xuemei Tang, Jia Yu, Qiang Fei, Wenneng Wu, Pei Li, Heng Luo   +6 more
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Synthesis and Estimation of the Insecticide and Antibacterial Activities for Some New Amide Derivatives

Indonesian Journal of Chemistry, 2023
In this work, new compounds of amide derivatives (C1-C3) were synthesized through the conversion reaction of p-chloroaniline to diazonium salt (B1), which reacts with aniline to form a new azo-compound (B3).
Zinah Hussein Ali, Dina Saleem, Abbas Khudhair Abbas, Baneen Salam Rasool, Mustafa Sabri Cheyad   +4 more
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Synthesis and RP-TLC lipophilicity evaluation of a novel fluocinolon acetonide soft drug derivative [PDF]

Kragujevac Journal of Science, 2016
Cortienic acid was obtained by periodic acid oxidation of fluocinolone acetonide, whereas corresponding amide was synthesized from the cortienic acid and ethyl ester of b-alanine by dicyclohexylcarbodiimide - hydroxybenzotriazole coupling procedure ...
Dobričić Vladimir, Vladimirov Sote, Čudina Olivera   +2 more
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Synthesis of Functionalized N-(4-Bromophenyl)furan-2-carboxamides via Suzuki-Miyaura Cross-Coupling: Anti-Bacterial Activities against Clinically Isolated Drug Resistant A. baumannii, K. pneumoniae, E. cloacae and MRSA and Its Validation via a Computational Approach

Pharmaceuticals, 2022
N-(4-bromophenyl)furan-2-carboxamide (3) was synthesized by the reaction furan-2-carbonyl chloride (1) and 4-bromoaniline (2) in the presence of Et3N in excellent yields of 94%.
Ayesha Siddiqa, Muhammad Zubair, Muhammad Bilal, Nasir Rasool, Muhammad Usman Qamar, Aqsa Khalid, Gulraiz Ahmad, Muhammad Imran, Sajid Mahmood, Ghulam Abbas Ashraf   +9 more
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Progress in C-C and C-Heteroatom Bonds Construction Using Alcohols as Acyl Precursors

Molecules, 2022
Acyl moiety is a common structural unit in organic molecules, thus acylation methods have been widely explored to construct various functional compounds.
Feng Zhao, Bin Tan, Qing Li, Qi Tan, Huawen Huang   +4 more
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Crystal structure of 2-(4-chlorobenzamido)benzoic acid

Acta Crystallographica Section E: Crystallographic Communications, 2015
In the title molecule, C14H10ClNO3, the amide C=O bond is anti to the o-carboxy substituent in the adjacent benzene ring, a conformation that facilitates the formation of an intramolecular amide-N—H...O(carbonyl) hydrogen bond that closes an S(6) loop ...
Rodolfo Moreno-Fuquen, Vanessa Melo, Javier Ellena   +2 more
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Synthesis of Gibberellic Acid Derivatives and Their Effects on Plant Growth

Molecules, 2017
A series of novel C-3-OH substituted gibberellin derivatives bearing an amide group were designed and synthesized from the natural product gibberellic acid (GA3).
Hao Tian, Yiren Xu, Shaojin Liu, Dingsha Jin, Jianjun Zhang, Liusheng Duan, Weiming Tan   +6 more
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Self-Assembled Fluorinated Organogelators for Surface Modification

Applied Sciences, 2012
A new class of alkyl- and perfluoroalkyl-containing urea and amide derivatives was synthesized from amino acid derivatives. Most of these compounds showed excellent gelation behavior in organic solvents at low concentrations.
Anilkumar Raghavanpillai, Vincent A. Franco   +1 more
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N,N-Diethyl-3-methylbenzamide

Molbank, 2022
The development of new techniques for the preparation of organic compounds is important, with catalytic processes being key to this innovation. The development of copper-based metal-organic frameworks to promote oxidative couplings has allowed the ...
María Albert-Soriano, Isidro M. Pastor
doaj   +1 more source