Results 51 to 60 of about 473,188 (208)

Amide-functionalized 1,2,4-Triazol-5-amines as Covalent Inhibitors of Blood Coagulation Factor XIIa and Thrombin

, 2022
To counteract thrombosis, new safe and efficient antithrombotics are required. We herein report the design, synthesis, and biological activity of a series of amide-functionalized acylated 1,2,4-triazol-5-amines as selective inhibitors of blood ...
Catharina Erbacher (14195802), Dmitrii V. Kalinin (5828132), Uwe Karst (1517185), Wolfgang Dörner (9260411), Constantin G. Daniliuc (1301925), Antti Poso (1760140), Lukas Imberg (9550718), Simon Platte (14195799), Svetlana A. Kalinina (4538362)   +8 more
core   +2 more sources

N-(2,4-Difluorophenyl)-2-fluorobenzamide

Molbank
The title compound N-(2,4-difluorophenyl)-2-fluorobenzamide (Fo24) was synthesized in high yield (1.09 g; 87%) using standard synthetic procedures from the condensation reaction of 2-fluorobenzoyl chloride with 2,4-difluoroaniline.
Niall Hehir, John F. Gallagher
doaj   +1 more source

Evaluation of the Inhibitory Effects of Pyridylpyrazole Derivatives on LPS-Induced PGE₂ Productions and Nitric Oxide in Murine RAW 264.7 Macrophages

Molecules, 2021
A series of thirteen triarylpyrazole analogs were investigated as inhibitors of lipopolysaccharide (LPS)-induced prostaglandin E2 (PGE2) and nitric oxide (NO) production in RAW 264.7 macrophages.
Mahmoud M. Gamal El-Din, Mohammed I. El-Gamal, Young-Do Kwon, Su-Yeon Kim, Hee-Soo Han, Sang-Eun Park, Chang-Hyun Oh, Kyung-Tae Lee, Hee-Kwon Kim   +8 more
doaj   +1 more source

Preparation and Characterization of Amide-Containing Polyimide Films with Enhanced Tribopositivity for Triboelectric Nanogenerators to Harvest Energy at Elevated Temperatures

Nanoenergy Advances
As triboelectric nanogenerator (TENG) technology continue to evolve, its application in harsh environments has increasingly captivated the interest of researchers.
Zhen Pan, Shunqi Yuan, Yan Zhang, Xi Ren, Zhibin He, Zhenzhong Wang, Shujun Han, Yuexin Qi, Haifeng Yu, Jingang Liu   +9 more
doaj   +1 more source

Fluorescence Spectroscopy of Enantiomeric Amide Compounds Enforced by Chiral Light

Applied Sciences, 2021
Chirality, the absence of mirror symmetry, governs behavior in most biologically important molecules, thus making the chiral recognition of great importance in the pharmaceutical and agrochemical industries, as well as medicine.
Alessandro Belardini, Emilija Petronijevic, Ramin Ghahri, Daniele Rocco, Fabiana Pandolfi, Concita Sibilia, Leonardo Mattiello   +6 more
doaj   +1 more source

Synthesis of 6- or 8-Carboxamido Derivatives of Imidazo[1,2-a]pyridines via a Heterogeneous Catalytic Aminocarbonylation Reaction

Molecules
Imidazo[1,2-a]pyridines and especially their amide derivatives exhibit a wide range of favourable pharmacological properties. In this work, Pd-catalysed carbonylation was used for the first time for the introduction of the carboxamide moiety into ...
Enikő Nagy, Attila Máriás, Margit Kovács, Rita Skoda-Földes   +3 more
doaj   +1 more source

Amide-Functionalized Polyolefins and Facile Post-Transformations

Direct copolymerization of olefins with polar monomers to produce functionalized polyolefins has attracted much attention; however, highly efficient incorporation of amide functions into polyolefins is a long-standing challenge because the amide function
Yixin Zhang (173038), Lei Cui (165714), Zhongbao Jian (1645531), Kangkang Li (1664689)   +3 more
core   +1 more source

Amide-Stabilized, Diamagnetic Chromium(II) Nitrosyl Complexes¹

, 2016
Treatment of Cr(NO)(NiPr2)3 with 2 equiv of PhCO2H affords Cr(NO)(NiPr2)(O2CPh)2 (1) in good yields. Reaction of CpNa·DME with 1 produces CpCr(NO)(NiPr2)(OC(O)Ph) (2), which subsequently yields a series of 18-valence-electron (18e) complexes, CpCr(NO ...
Eric W. Jandciu (3086433), Steven J. Rettig (2092000), Peter Legzdins (1406356), Jane Kuzelka (2525995), Kevin M. Smith (1316334)   +4 more
core   +3 more sources

Efficient Straightforward Synthesis of Amidopiperazinophanes as Versatile Novel Supramolecular Scaffolds

SynOpen, 2019
A simple one-pot synthesis of amidopiperazinophanes with a combination of electron-deficient amide groups and electron-rich alkyne and piperazine functionalities has been achieved by using multicomponent reaction (MCR) methodology with the Mannich ...
Ayyavu Thirunarayanan, Sivasamy Selvarani, Gracia Francisco, Perumal Rajakumar   +3 more
doaj   +1 more source

Adsorption of alkyl amides: monolayer structures and mixing behaviour [PDF]

, 2011
In this work monolayers of alkyl amides adsorbed on a graphite surface have been successfully identified and investigated using a combination of synchrotron X-ray and neutron diffraction and Differential Scanning Calorimetry (DSC).

core   +2 more sources