Results 71 to 80 of about 463 (98)

Backbone nitrogen substitution restricts the conformation of glycine residues in β-turns. [PDF]

Chem Commun (Camb)
Gu F, Thomas D, Newberry RW.
europepmc   +1 more source

Atazanavir-Loaded Crosslinked Gamma-Cyclodextrin Nanoparticles to Improve Solubility and Dissolution Characteristics. [PDF]

Turk J Pharm Sci, 2022
Dhabliya D, Khan SAQ, Umate M, Raut B, Singhavi D.   +4 more
europepmc   +1 more source

Recent applications of computational methods to allosteric drug discovery. [PDF]

Front Mol Biosci, 2022
Govindaraj RG, Thangapandian S, Schauperl M, Denny RA, Diller DJ.   +4 more
europepmc   +1 more source

Azapeptides with unique covalent warheads as SARS-CoV-2 main protease inhibitors. [PDF]

Antiviral Res
Khatua K, Alugubelli YR, Yang KS, Vulupala VR, Blankenship LR, Coleman D, Atla S, Chaki SP, Geng ZZ, Ma XR, Xiao J, Chen PH, Cho CD, Sharma S, Vatansever EC, Ma Y, Yu G, Neuman BW, Xu S, Liu WR.   +19 more
europepmc   +1 more source

Azapeptide-Based SARS-CoV-2 Main Protease Inhibitors: Design, Synthesis, Enzyme Inhibition, Structural Determination, and Antiviral Activity. [PDF]

J Med Chem
Flury P, Vishwakarma J, Sylvester K, Higashi-Kuwata N, Dabrowska AK, Delgado R, Cuell A, Basu R, Taylor AB, de Oliveira EG, Magalhães Serafim MS, Qiao J, Chen Y, Yang S, O'Donoghue AJ, Mitsuya H, Gütschow M, Laufer SA, Müller CE, Harris RS, Pillaiyar T.   +20 more
europepmc   +1 more source

Microparticles of Sericin-Dextran Conjugate for Improving the Solubility of Antiviral Drug. [PDF]

J Funct Biomater, 2023
Chen S, Feng X, Li X, Liu M, Gao W, Miao Q, Wu H.   +6 more
europepmc   +1 more source

Inhibitors of Proteinases as Potential Anti-Cancer Agents [PDF]

, 2011
Karolina Gluza, Paweł Kafarski
core   +1 more source

Novel inhibitors and activity-based probes targeting serine proteases. [PDF]

Front Chem, 2022
Ferguson TEG, Reihill JA, Martin SL, Walker B.   +3 more
europepmc   +1 more source

Design, Synthesis, and Evaluation of Aza-Peptide Michael Acceptors as Human 20S Proteasome Inhibitors: Extension to the Prime Site

ACS Omega
Sarah E. Border, Leilani M. Lotti Diaz, Rasmiah Amer, Abigail M. Noonchester, Kayla S. Kucway, Michael Fleisher, Joseph P. Fernandez, Alex R. Lovins, Thomas S. Corrigan, Ana K. Serrano, Conor R. Caffrey, Anthony J. O’Donoghue, Don M. Benson, Christopher M. Hadad, Özlem Doğan Ekici   +14 more
doaj   +1 more source

Recent Patents and FDA-Approved Drugs Based on Antiviral Peptides and Other Peptide-Related Antivirals. [PDF]

Int J Pept Res Ther, 2023
Mousavi Maleki MS, Sardari S, Ghandehari Alavijeh A, Madanchi H.   +3 more
europepmc   +1 more source