Results 201 to 210 of about 16,265 (239)
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Alkylating benzamides with melanoma cytotoxicity
Melanoma Research, 2004Radioiodinated N-(2-(diethylamino)ethyl)benzamides have recently been discovered as selective agents for melanotic melanoma and are used for scintigraphic imaging in nuclear medicine. Owing to the high binding capacity, benzamide derivatives conjugated with alkylating cytostatics were synthesized and tested for their potential for targeted drug ...
Markus, Wolf +6 more
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Chemical Synthesis of Benzamide Riboside
Current Medicinal Chemistry, 2002The C-glycosidic nicotinamide riboside analogue (1) was prepared by reaction of ribonolactone 16 with the lithiated 2-oxazoline 13 followed by triethylsilane reduction of the hemiacetal 17 to the tetrahydrofurane 18. Cleavage of the oxazoline group in 20 to the acid 21, conversion of the acid chloride 22 to the amide 23, and hydrogenative debenzylation
K, Krohn, H, Dörner, M, Zukowski
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Benzamides and cholinesterases.
Research communications in chemical pathology and pharmacology, 1987At certain doses metoclopramide (MT), sulpiride and bromopride produce anti-cholinesterase effects as shown by studies on the serum and erythrocyte cholinesterases of the rabbit and the dog, and by those on the hypotensive effect of ACh incubated with rabbit serum in the presence or absence of MT. The anti-cholinesterase effect of MT was more intensive
VACCA C +3 more
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Photocatalytic modifications of benzamides
2022Benzamide derivatives are highly prevalent in biologically active compounds, including approved and investigational drugs of diverse mechanism of action. They have also been exploited as radiotracers for melanoma imaging and as chromophores for stereochemical studies by circular dichroism.
Maciej Giedyk, Agnieszka Kamińska
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Silicon in benzamide directed ortho metalation. Formation and reactions of benzamide benzynes
Tetrahedron Letters, 1984Abstract 2-Trimethylsilyl-3-triflyl benzamide 3 , undergoes fluoride-mediated 1,2-elimination to give the benzyne intermediate 4 which is trapped by cycloaddition ( 5 ), and nucleophilic reactions ( 6 ).
K. Shankaran, V. Snieckus
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Pigment & Resin Technology, 1999
Aqueous sodium chloride solution, containing benzamide was electrolysed (pH = 2), using platinised titanium anode and graphite cathode. The filtrate of the reaction mixture (pH = 4.5) was diazotised and coupled with α‐naphthol in NaOH and also with β‐naphthol in NaOH. Dyes were produced.
Susai Rajendran +2 more
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Aqueous sodium chloride solution, containing benzamide was electrolysed (pH = 2), using platinised titanium anode and graphite cathode. The filtrate of the reaction mixture (pH = 4.5) was diazotised and coupled with α‐naphthol in NaOH and also with β‐naphthol in NaOH. Dyes were produced.
Susai Rajendran +2 more
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L'Encephale, 1976
The comparison of the therapeutic effects of three molecules belonging to the substituted benzamide family allows the following observations: --the three products are generally well tolerated by the organism; --at sufficient doses they act as a major tranquilizers: -sulpiride is chiefly a disinhibitor but also has antipsychotic properties; -sultopride ...
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The comparison of the therapeutic effects of three molecules belonging to the substituted benzamide family allows the following observations: --the three products are generally well tolerated by the organism; --at sufficient doses they act as a major tranquilizers: -sulpiride is chiefly a disinhibitor but also has antipsychotic properties; -sultopride ...
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Structure of a benzamide derivative
Acta Crystallographica Section C Crystal Structure Communications, 1985Amino-5-chloro-2-methoxy-N- { 2-(N- (p- ro ethoxybenzyl)methylamino )- 1,1 -dimethylethyl } benz- amide, C21H28CIN303, M r = 405.93, monoclinic, P21/c, a = 6.144 (I), b = 26.512 (2), c = 13.741 (2) A, fl=94.76(1) °, V= 2230.5 (5) A3, Z=4, D_= 1.21, D x = 1.209 gcm -3, /),(Mo Ka) = 0.71073 ~, It = 1.92cm -I, F(000)=864, room temperature, R= 0.076 for ...
T. Furuya +3 more
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Zeitschrift für anorganische und allgemeine Chemie, 2008
Jürgen Thun, Josef Breu
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Jürgen Thun, Josef Breu
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