Novel piperazine-triazole hybrids as PTP1B and alpha-amylase inhibitors: synthesis, biological evaluation and computational validation through network pharmacology, molecular docking, MD simulations, DFT and MMPBSA analysis. [PDF]
Haroon M, Kamal S, Mansha A, Zahoor AF.
europepmc +1 more source
Development of a Second-Generation RARα Selective Antagonist as an Orally Bioavailable, Effective, Safe, and Reversible Male Contraceptive. [PDF]
Shi R +8 more
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Design, characterization, DFT studies, and molecular docking of new benzofuran-pyrazol-acrylamide hybrids as insecticidal agents against Spodoptera littoralis and Tribolium castaneum. [PDF]
El-Bana GG +5 more
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Development of Bioisosteres of Iboga Alkaloids: A Step-Economical Synthesis to Enhance the Antinociceptive and Anxiolytic Activity with Neuroprotective Effects. [PDF]
Gupta A +9 more
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Total Synthesis of the Oligostilbenes Anigopreissin A and Fuliginosin A. [PDF]
Ramos Orea A +3 more
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Synthesis of benzofuran-based benzimidazole compounds andinvestigation of their antidiabetic effects
Bu tez çalışması kapsamında öncelikle 2-aril-4,6-dimetil ve 2-aril-4,6-dimetoksi benzofuran bileşiklerinin sentezlenmiş daha sonra bu sentezlenen öncü bileşikler Vilsmeier-Haack reaksiyonuna tabi tutularak seçici olarak C3 ve C7 pozisyonlarına aldehit ...
Ocak, İclal
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5-(Benzofuran-2-yl)-3-(2-chloro-4-fluorobenzyl)-1,3,4-oxadiazol-2(3H)-one (GM-90663) Alleviates Dravet Syndrome via Inhibiting Monoamine Oxidase Activity. [PDF]
Hwang KS +16 more
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Benzofuran compound from <i>Sophora tonkinensis Gagnep</i> suppresses nasopharyngeal carcinoma growth via PI3K/AKT/mTOR pathway: evidence from molecular dynamics simulation and <i>in vitro</i> experiments. [PDF]
Wu P +11 more
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Naphthalimide Derivatives with Extended Heterocyclic Systems-Synthesis, Spectral and Sensing Properties. [PDF]
Manov H +7 more
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