New N-phenylpyrrolamide inhibitors of DNA gyrase with improved antibacterial activity. [PDF]
Cotman AE +19 more
europepmc +1 more source
Signal Propagation in the ATPase Domain of Mycobacterium tuberculosis DNA Gyrase from Dynamical-Nonequilibrium Molecular Dynamics Simulations. [PDF]
Kamsri B +9 more
europepmc +1 more source
Identification of Anti-Tuberculosis Drugs Targeting DNA Gyrase A and Serine/Threonine Protein Kinase PknB: A Machine Learning-Assisted Drug-Repurposing Approach. [PDF]
Lee D +6 more
europepmc +1 more source
Membrane translocation and refolding mitochondrial proteins [PDF]
Hartl, Franz-Ulrich +2 more
core
Characterization of a prokaryotic topoisomerase I activity in chloroplast extracts of maize [PDF]
Siedlecki, Janusz +2 more
core
New N-amino-5-cyano-6-pyridones as antimicrobial small molecules endowed with DNA gyrase a inhibitory activity: design, one-pot synthesis, biological assessment and in silico insights. [PDF]
Kamaly OA +5 more
europepmc +1 more source
Ligand-Based Virtual Screening for Discovery of Indole Derivatives as Potent DNA Gyrase ATPase Inhibitors Active against Mycobacterium tuberculosis and Hit Validation by Biological Assays. [PDF]
Pakamwong B +18 more
europepmc +1 more source
Two classes of DNA gyrase inhibitors elicit distinct evolutionary trajectories toward resistance in gram-negative pathogens. [PDF]
Leyn SA +5 more
europepmc +1 more source
Dynamic Profiling and Binding Affinity Prediction of NBTI Antibacterials against DNA Gyrase Enzyme by Multidimensional Machine Learning and Molecular Dynamics Simulations. [PDF]
Kokot M, Minovski N.
europepmc +1 more source

