Design and Synthesis of Structurally Modified Analogs of 24Z-Isomasticadienonic Acid with Enhanced Anti-Proliferative Activity [PDF]
Τriterpenic acids represent a prominent class of bioactive compounds, with a wide range of biological properties, including anti-inflammatory, antiviral, and anticancer effects. Among them, 24Z-isomasticadienonic acid (IMNA), a major constituent of Chios
Panagiota Stamou +5 more
doaj +2 more sources
Synthesis Characterization of Some New Heterocyclic Compounds Containing1, 3-Oxazepine Ring [PDF]
تم تحضیر سلسلة من مشتقات 1, 3 - الاوکسازبین من خلال خطوتین الاول: یتضمن تحضیر مشتقات الایمین (A7-A1) من تفاعل 4 - هیدروکسی بنزالدیهاید مع امینات معوضة مختلفة وباستخدام حامض الخلیک الثلجی.
Jawdat H. Abdul – Wahid +2 more
doaj +1 more source
Heterocyclic compounds are one of the main groups of organic compounds possessing wide range of applications in various areas of science and their derivatives are present in many bioactive structures. They display a wide variety of biological activities.
Benas Balandis +2 more
doaj +1 more source
The purpose of this research is to prepare new vanillic acid derivatives with 1,2,4-triazole-3-thiol heterocyclic ring and evaluate their antimicrobial activity in a preliminary assessment.
Noor Ali Sabzi, May Mohammed Jawad
doaj +1 more source
Preparation and diagnosis some heterocyclic compounds that derived from 1,3,4 – Thiadiazole compound derived from 1,3,4 – Thiadiazole compound [PDF]
This search included synthesis of some heterocyclic compounds devired from 1,3,4- thiadiazol ring ,such as thaiazolidin -4-one substituents Azetidine -3- one and Azo dyes.
Ayad S. H. AL-Maaini Nazhan.KA AL-Luhiby
doaj +1 more source
Synthesis and Reactivity of 3H-1,2-dithiole-3-thiones
3H-1,2-Dithiole-3-thiones are among the best studied classes of polysulfur-containing heterocycles due to the almost explosive recent interest in these compounds as sources of hydrogen sulfide as an endogenously produced gaseous signaling molecule.
Oleg A. Rakitin
doaj +1 more source
Methods for the synthesis of polyhydroxylated piperidines by diastereoselective dihydroxylation: Exploitation in the two-directional synthesis of aza-C-linked disaccharide derivatives [PDF]
Background: Many polyhydroxylated piperidines are inhibitors of the oligosaccharide processing enzymes, glycosidases and glycosyltransferases. Aza-C-linked disaccharide mimetics are compounds in which saturated polyhydroxylated nitrogen and oxygen ...
Adam Nelson +8 more
core +3 more sources
Synthesis, characterization, and antimicrobial evaluation of new Schiff bases derived from vanillic acid conjugated to heterocyclic 4H-1,2,4-triazole-3-thiol [PDF]
A multistep synthesis was established for the preparation of a new vanillic acid-1, 2, 4-1triazole-3-thiol conjugate (4). Finally, several aromatized aldehydes reacted with compound (4) to produce Schiff bases derivatives (5–11).
Noor Ali Hussein Sabzi +1 more
doaj +3 more sources
1,3-Oxazepane-4,7-Diones Compounds: 1Hand 13CNMR High-Resolution Spectroscopy (1D and 2D) [PDF]
“Oxazepine” refers to any seven-membered ring containing an oxygen and nitrogen atom. The 1,3-oxazepine is a branch of many types of the heterocyclic oxazepine [1–7].
Abdul Karim , Talaq Mohammad +2 more
core +1 more source
Microwave-assisted syntheses of novel ring d-condensed 2-pyrazolines in the estrone series were efficiently carried out from steroidal α,β-enones and hydrazine derivatives. The ring-closure reaction of 16-benzylidene estrone 3-methyl ether with
Gergő Mótyán +3 more
doaj +1 more source

