Results 161 to 170 of about 57,473 (326)

Effect of Ions and Sequence Variants on the Antagonist Binding Properties of the Histamine H₁ Receptor. [PDF]

Int J Mol Sci, 2022
Conrad M, Söldner CA, Sticht H.
europepmc   +1 more source

Suppression of Histamine Signaling by Probiotic Lac-B: a Possible Mechanism of Its Anti-allergic Effect

Journal of Pharmacological Sciences, 2008
It has been shown that probiotic bacteria are effective for the treatment of allergic diseases. As histamine plays a central role in allergic diseases, it is possible that probiotic bacteria affect the allergy-related histamine signaling.
Shrabanti Dev, Hiroyuki Mizuguchi, Asish K. Das, Chiyo Matsushita, Kazutaka Maeyama, Hayato Umehara, Takayuki Ohtoshi, Jun Kojima, Kiyotaka Nishida, Kunihiko Takahashi, Hiroyuki Fukui   +10 more
doaj  

Optimization of Peptide Linker-Based Fluorescent Ligands for the Histamine H₁ Receptor. [PDF]

J Med Chem, 2022
Kok ZY, Stoddart LA, Mistry SJ, Mocking TAM, Vischer HF, Leurs R, Hill SJ, Mistry SN, Kellam B.   +8 more
europepmc   +1 more source

Stimulatory (H1) and Inhibitory (H2) Histamine Receptors in Gallbladder Muscle

, 1977
Daniel Waldman, Alvin M. Zfass, G.M. Makhlouf   +2 more
openalex   +1 more source

STUDIES OF HISTAMINE, H1 AND H2 RECEPTORS IN BRONCHOCONSTRICTION

The KITAKANTO Medical Journal, 1990
To clarify the roles of H1 and H2 receptors in the airways of asthmatic patients, we studied the effects of the administration of a histamine H1 receptor antagonist, an H2 receptor antagonist and a combination of both on bronchial constriction induced by histamine inhalation and allergen inhalation in patients with asthma.We also examined the effects ...
openaire   +3 more sources

Quantitation of Phototoxic Hyperemia and Permeability to Protein: II. Inihibition by Histamine (H1 and H2) Receptor Antagonists in Mouse Skin

, 1980
Lawrence W. Argenbright, P. Donald Forbes, Gwendolyn J. Stewart   +2 more
openalex   +1 more source

Exploring the Effect of Cyclization of Histamine H₁ Receptor Antagonists on Ligand Binding Kinetics. [PDF]

ACS Omega, 2021
Wang Z, Bosma R, Kuhne S, van den Bor J, Garabitian W, Vischer HF, Wijtmans M, Leurs R, de Esch IJP.   +8 more
europepmc   +1 more source

Histamine H1 receptor in endothelium and smooth muscle of guinea pig aorta

, 1986
Michihiro Hide, Hiroyuki Fukui, Takehiko Watanabe, Shoso Yamamoto, Hiroshi Wada   +4 more
openalex   +1 more source

Pharmacology of Antihistamines

World Allergy Organization Journal, 2011
This article reviews the molecular biology of the interaction of histamine with its H1-receptor and describes the concept that H1-antihistamines are not receptor antagonists but are inverse agonists i.e.
Diana S Church, MD, Martin K Church, PhD
doaj  

BRET-Based Biosensors to Measure Agonist Efficacies in Histamine H₁ Receptor-Mediated G Protein Activation, Signaling and Interactions with GRKs and β-Arrestins. [PDF]

Int J Mol Sci, 2022
Verweij EWE, Bosma R, Gao M, van den Bor J, Al Araaj B, de Munnik SM, Ma X, Leurs R, Vischer HF.   +8 more
europepmc   +1 more source