Results 201 to 210 of about 45,597 (259)

Novel machine learning approach toward classification model of HIV-1 integrase inhibitors [PDF]

Tieu-Long Phan, Hoang-Son Lai Le, Gia-Bao Truong, The-Chuong Trinh, Van-Thinh To, Phuoc-Chung Van Nguyen, Thanh-An Pham, Tuyen Ngoc Truong   +7 more
openalex   +1 more source

858: Integrase inhibitor versus protease inhibitor (PI)-based antiretroviral therapy (ART) in late pregnancy and rapid HIV viral load reduction in ART naïve patients: Cost effectiveness analysis [PDF]

, 2018
Ahizechukwu C. Eke, Kelly E. Dooley, Jeanne S. Sheffield   +2 more
openalex   +1 more source

5-Hydroxypyrido[2,3-b]pyrazin-6(5H)-one derivatives as novel dual inhibitors of HIV-1 reverse transcriptase-associated ribonuclease H and integrase

, 2018
Lin Sun, Ping Gao, Guanyu Dong, Xujie Zhang, Xiqiang Cheng, Xiao Ding, Xueshun Wang, Dirk Daelemans, Erik De Clercq, Christophe Pannecouque, Luis Menéndez‐Arias, Peng Zhan, Xinyong Liu   +12 more
openalex   +2 more sources

Design, synthesis and biological evaluation of (E)-3,4-dihydroxystyryl 4-acylaminophenethyl sulfone, sulfoxide derivatives as dual inhibitors of HIV-1 CCR5 and integrase

, 2016
Yixing Sun, Weisi Xu, Ningning Fan, Xuefeng Sun, Xianling Ning, Liying Ma, Junyi Liu, Xiaowei Wang   +7 more
openalex   +1 more source

Elucidating the Mechanism by Which HIV-1 Nucleocapsid Mutations Confer Resistance to Integrase Strand Transfer Inhibitors [PDF]

Yuta Hikichi, Ryan C. Burdick, Sean C. Patro, Si-Yuan Ding, Brian T. Luke, Erin Clark, Sherimay D. Ablan, Xiaolin Wu, Vinay K. Pathak, Eric O. Freed   +9 more
openalex   +1 more source

The Road to HIV-1 Integrase Inhibitors: The Case for Supporting Basic Research

, 2014
Robert Craigie
openalex   +1 more source

Molecular dissection of an inhibitor targeting the HIV integrase dependent preintegration complex nuclear import. [PDF]

Cell Microbiol, 2019
Wagstaff KM, Headey S, Telwatte S, Tyssen D, Hearps AC, Thomas DR, Tachedjian G, Jans DA.   +7 more
europepmc   +1 more source

Structural basis for the potent inhibition of the HIV integrase-LEDGF/p75 protein–protein interaction

, 2017
Sergio R. Ribone, Mario A. Quevedo
openalex   +2 more sources

Real-world Prevalence of Nonintegrase INSTI Resistance-Associated Mutations and Virological Outcomes in People Who Have Recently Acquired HIV-1 in the United Kingdom. [PDF]

J Infect Dis
Kelly C, Lester JS, Bradshaw D, Bibby DF, Mohamed H, Murphy G, Brown A, Sabin C, Geretti AM, Mbisa JL.   +9 more
europepmc   +1 more source

Pharmacophore‐Based Discovery of Small‐Molecule Inhibitors of Protein–Protein Interactions between HIV‐1 Integrase and Cellular Cofactor LEDGF/p75

, 2009
Laura De Luca, Maria Letizia Barreca, Stefania Ferro, Frauke Christ, Nunzio Iraci, Rosaria Gitto, Anna Maria Monforte, Zeger Debyser, Alba Chimirri   +8 more
openalex   +2 more sources