Results 101 to 110 of about 7,519 (213)

Improved synthesis of 6-[(ethylthio)methyl]-1H-indazole

, 2015
cited By 2International audienceIn the improved synthesis of 6-[(ethylthio)methyl]-1H-indazole (5), the mesylate intermediate is replaced by the bromide derivative, which increases the overall yield (six steps) by a factor of ...
Stefak, Roman, Rapenne, Gwénaël, Sirven, Agnès M.   +2 more
core   +1 more source

Regioselective synthesis of novel substituted indazole-5,6-diamine derivatives

, 2011
International audienceThe synthesis of a series of novel indazole-5,6-diamine derivatives is described. This indazole ring system was incorporated in an octahydropyrrolo[3,4-b]phenazine scaffold and was diversely and regioselectively substituted on the ...
Saugues, Emmanuelle, Anizon, Fabrice, Gavara, Laurent, Moreau, Pascale   +3 more
core   +1 more source

New Syntheses of Indazole and 2-Substituted Indazoles. [PDF]

Acta Chemica Scandinavica, 1975
Jan M. Bakke, Kjell A. Skjervold, Birgitta Gotthammar   +2 more
openaire   +1 more source

1-Allyl-3-chloro-5-nitro-1H-indazole

, 2013
In the title compound, C10H8ClN3O2, the indazole ring system makes a dihedral angle of 7.9 (3)° with the plane through the nitro group. The allyl group is rotated out of the plane of the indazole ring system [N—N—C—C torsion ...
El Mostapha Rakib, Hakima Chicha, Mohamed Saadi, Domenico Spinelli, Lahcen El Ammari   +4 more
core   +1 more source

Synthesis and diversification of SuFEx-active 2<i>H</i>-indazoles from azobenzenes and ethenesulfonyl fluoride. [PDF]

RSC Adv
Rajaka L, Woo H, Jung M, Jang C, Kim S, Lee J, Kim S, Han S, Bae HY, Han SH.   +9 more
europepmc   +1 more source

Structure-activity profiling of indazole-based derivatives as spinster homolog 2 (Spns2)-dependent S1P release inhibitors. [PDF]

Bioorg Med Chem Lett
Hernandez M, Hawkins DJ, Kharel Y, Huang T, Prendergast AD, Brown AM, Lynch KR, Santos WL.   +7 more
europepmc   +1 more source

Solid state forms of 2-{4-[(3S)-piperidin-3-yl]phenyl}-2H-indazole-7-carboxamide salts and processes for preparation thereof [PDF]

The present invention provides solid state forms of 2-{4-[(3S)-piperidin-3-yl]phenyl}-2H-indazole-7-carboxamide salts and processes for preparation thereof.
, Srinivasan Thirumalai Rajan, Sagyam Rajeshwar Reddy, Kammari Bal Raju, Garai Abhijit, Padigapaty Shiva Reddy, MSN Laboratories Private Limited, R&D Center, Hyderabad, India.
core  

Activating Photoreaction of Indazole Metastable-State Photoacid through Two-Photon Excitation. [PDF]

J Phys Chem Lett
Ma YZ, Liyanage P, Liao Y.
europepmc   +1 more source

N-(1H-Indazolyl) Aryl Sulfonamide Hybrids as Potential Dihydropteroate Synthase Inhibitors: In Vitro Antibacterial Activity Against Escherichia coli and Staphylococcus aureus and Computational Modeling. [PDF]

Chem Biodivers
Boudza R, Elandaloussi F, Boujdi K, Segura-Garcia J, Brahmi NE, Kazzouli SE, Moukadiri I, Maicas S, Bounou S.   +8 more
europepmc   +1 more source

Advances in N- and S-Heterocycles as c-Jun-N-Terminal Kinase 3 Inhibitors for Alzheimer's Disease Treatment. [PDF]

Drug Dev Res
Yadav P, Mishra D, Singh R.
europepmc   +1 more source