Results 91 to 100 of about 4,776 (179)

<i>N</i>-Heterocyclic Olefins of Pyrazole and Indazole. [PDF]

Org Lett
Zhu B, Woyciechowski R, Hübner EG, Lederle F, Schmidt A.   +4 more
europepmc   +1 more source

SAR Studies around the SULT1A1-Activated Alkylator YC-1 as Cytotoxic Agents against Biliary Tract Cancer Cells. [PDF]

J Med Chem
Kong K, Zhao W, Shrimp JH, Vava M, Sinha R, Sharma S, Lee TD, Roth JS, Lee OW, Lewis D, Kearney SE, Rohde JM, Davis MI, Shah P, Wang AQ, Xu X, Shi L, Shen M, Boxer MB, Bardeesy N, Hall MD, Patnaik S.   +21 more
europepmc   +1 more source

Novel Substituted Indazoles as Small Molecule-Based Inhibitors of KRAS Proteins. [PDF]

ACS Med Chem Lett
Rong J, Liang SH.
europepmc   +1 more source

Simulation of the Metabolism of New Psychoactive Substances Using Electrochemistry-Mass Spectrometry: Introducing an Innovative Software Tool for Rapid Data Evaluation. [PDF]

Drug Test Anal
Wesner M, Heuckeroth S, Pütz M, Karst U.   +3 more
europepmc   +1 more source

Design, synthesis, and antiproliferative activity of new 5-ethylsulfonyl-indazole-3-carbohydrazides as dual EGFR/VEGFR-2 kinases inhibitors. [PDF]

J Enzyme Inhib Med Chem
Al-Wahaibi LH, Abou-Zied HA, Mahmoud MA, Youssif BGM, Bräse S, Rabea SM.   +5 more
europepmc   +1 more source

In vitro CB₁ receptor activity of halogenated indazole synthetic cannabinoid receptor agonists. [PDF]

Arch Toxicol
Green H, McKenzie C, Hamra E, Rautio T, Wu X, Juneskog E, Sandblom R, Monti MC, Persson M, Norman C.   +9 more
europepmc   +1 more source

The Effect of <i>N</i>-Alkyl Azole Difluorination on Molecular Properties Relevant for Compound Optimization: A Comparative Study. [PDF]

ACS Med Chem Lett
Herrick RM, Green SA, Rich S, Grandner JM, Huard K, Altman RA.   +5 more
europepmc   +1 more source

Study on Phase I Metabolic Processes and Metabolite Biomarker Identification of Synthetic Cannabinoids 5F-ADB-PINACA and 5F-ADBICA in Human Liver Microsomes and Zebrafish Model. [PDF]

Molecules
Li H, Zheng H, Zhong S, Zhao Y, Lin J, Su H, Qian Z, Wang Y.   +7 more
europepmc   +1 more source

Synthetic cannabinoid receptor agonists containing silicon: exploring the metabolic pathways of ADMB- and Cumyl-3TMS-PrINACA in human urine specimens and post mortem material compared to in vitro and in silico data. [PDF]

Arch Toxicol
Zschiesche A, Carlier J, Pietsch J, Scheu M, Seibt J, Busardò FP, Auwärter V, Huppertz LM.   +7 more
europepmc   +1 more source

Arabidopsis P4-ATPases ALA1 and ALA7 Enhance Resistance to <i>Verticillium dahliae</i> via Detoxifying Vd-Toxins. [PDF]

Biology (Basel)
Wang F, Qiu M, Yao X, Li J, Ren H, Su M, Shen J, Li C, Jiang Q, Zhang Z, Li Y, Tang J, Li X, Fan Y, Pei Y.   +14 more
europepmc   +1 more source