Results 191 to 200 of about 2,808,349 (298)

Identification and Optimization of a Novel HIV-1 Integrase Inhibitor. [PDF]

ACS Omega, 2022
Adu-Ampratwum D, Pan Y, Koneru PC, Antwi J, Hoyte AC, Kessl J, Griffin PR, Kvaratskhelia M, Fuchs JR, Larue RC.   +9 more
europepmc   +1 more source

Safety and Pharmacokinetics of GSK364735, a Human Immunodeficiency Virus Type 1 Integrase Inhibitor, following Single and Repeated Administration in Healthy Adult Subjects [PDF]

, 2007
Y. Sunila Reddy, Sherene Min, Julie Borland, Ivy Song, Lin Jiang, Sandra M. Palleja, William T. Symonds   +6 more
openalex   +1 more source

Discovery and Preclinical Profiling of GSK3839919, a Potent HIV-1 Allosteric Integrase Inhibitor. [PDF]

ACS Med Chem Lett, 2022
Parcella K, Parcella K, Wang T, Eastman K, Zhang Z, Yin Z, Patel M, Tu Y, Zheng BZ, Walker MA, Saulnier MG, Frennesson D, Bowsher M, Gillis E, Peese K, Belema M, Cianci C, Dicker IB, McAuliffe B, Ding B, Falk P, Simmermacher J, Parker DD, Sivaprakasam P, Kish K, Lewis H, Hanumegowda U, Jenkins S, Kadow JF, Krystal M, Meanwell NA, Naidu BN.   +31 more
europepmc   +1 more source

Raltegravir: a potent and safe integrase inhibitor with a favourable impact on cardiovascular and liver profile [PDF]

, 2008
Francisco J. Blanco, Miguel Arredondo, Freddy Guevara, Carmen Garrido, Judit Morelló, Sonia Rodrı́guez-Nóvoa, Mònica Córdoba, Juan González‐Lahoz, Vincent Soriano   +8 more
openalex   +1 more source

Altered adipose tissue macrophage populations in people with HIV on integrase inhibitor-containing antiretroviral therapy. [PDF]

AIDS, 2022
Vakili S, Paneru B, Guerrier CM, Miller J, Baumrin E, Forrestel A, Lynn K, Frank I, Lo Re V, Collman RG, Hill DA.   +10 more
europepmc   +1 more source

Styrylquinolines, Integrase Inhibitors Acting Prior to Integration: a New Mechanism of Action for Anti-Integrase Agents

, 2004
Sabine Bonnenfant, Claire M. Thomas, Claudio Vita, Frédéric Subra, Eric Deprez, Fatima Zouhiri, Didier Desmaële, Jean d’Angelo, Jean François Mouscadet, Hervé Leh   +9 more
openalex   +1 more source

Mutations Associated with Failure of Raltegravir Treatment Affect Integrase Sensitivity to the Inhibitor In Vitro [PDF]

, 2008
Isabelle Malet, Olivier Delelis, Marc‐Antoine Valantin, Brigitte Montès, Cathia Soulié, Marc Wirden, Luba Tchertanov, Gilles Peytavin, Jacques Reynes, Jean‐François Mouscadet, Christine Katlama, Vincent Cálvez, Anne‐Geneviève Marcelin   +12 more
openalex   +1 more source

Changes in Body Mass Index with Longer-term Integrase Inhibitor Use: A Longitudinal Analysis of Data from the Randomized Trial to Prevent Vascular Events in Human Immunodeficiency Virus (REPRIEVE). [PDF]

Clin Infect Dis, 2023
Kileel EM, Malvestutto CD, Lo J, Fitch KV, Fichtenbaum CJ, Aberg JA, Zanni MV, Martinez E, Okeke NL, Kumar P, Joao E, Bares SH, Berrner D, Smieja M, Roa JC, McCallum S, Douglas PS, Ribaudo HJ, Grinspoon SK.   +18 more
europepmc   +1 more source

Integrase Inhibitor Use Associated with Weight Gain in Women and Incident Diabetes Mellitus. [PDF]

AIDS Res Hum Retroviruses, 2022
Asundi A, Olson A, Jiang W, Varshney SP, White LF, Sagar M, Lin NH.   +6 more
europepmc   +1 more source

Phenotypic analysis of HIV-1 E157Q integrase polymorphism and impact on virological outcome in patients initiating an integrase inhibitor-based regimen

Journal of Antimicrobial Chemotherapy, 2018
C. Charpentier, I. Malet, E. Andre-Garnier, A. Storto, L. Bocket, C. Amiel, L. Morand‐Joubert, C. Tumiotto, Thuy Nguyen, A. Maillard, A. Rodallec, M. Leoz, B. Montes, V. Schneider, J. Plantier, J. Dina, C. Pallier, A. Mirand, C. Roussel, A. Signori-Schmuck, S. Raymond, V. Calvez, C. Delaugerre, A. Marcelin, D. Descamps   +24 more
semanticscholar   +1 more source