The synthesis of 2‐methyl propellane and its conversion to various 1,2‐ and 1,2,3‐di‐ and trisubstituted bicyclopentanes is reported. Abstract Bicyclo[1.1.1]pentanes (BCPs) have emerged as isosteric replacements for mono‐ and para‐substituted benzene rings in medicinal and materials applications, involving substitution at the BCP bridgehead (1,3 ...
Sean R. Verschaeve +4 more
wiley +1 more source
Identification of epigenetic monotherapy candidates in taxane-resistant CRPC. [PDF]
Cevatemre B +3 more
europepmc +1 more source
Peer review of the pesticide risk assessment of the active substance proquinazid. [PDF]
European Food Safety Authority (EFSA) +47 more
europepmc +1 more source
On-Resin Synthesis and Late-Stage Functionalization of Macrocyclic Atosiban Mimetics via 5-Iodo-1,4-triazoles. [PDF]
Shepperson OA +4 more
europepmc +1 more source
Classification of Thyroid Peroxidase (TPO) Inhibitors Using Transfer Learning with SMILES Embeddings. [PDF]
Piir G +6 more
europepmc +1 more source
Discovery of Fused Isoquinolinone/Triazole as a Scaffold for Tankyrase and PARP Inhibition. [PDF]
Ouzounthanasis KA +8 more
europepmc +1 more source
An Organometallic [2]Catenane With Pt‒(di-NHC)‒Pt Units: A Topology-Driven Strategy for Enhanced Phosphorescence in Discrete Aggregates. [PDF]
Lu Y +5 more
europepmc +1 more source
Ketone Oximes as NO<sub>2</sub> Radical Precursors for Regioselective Iodo-Nitrosylative Cyclization of Unactivated 1,6-Enynes. [PDF]
Mutra MR +4 more
europepmc +1 more source
Photocatalytic <i>In Situ</i> Activation of Bench-Stable Saccharides: A General Synthetic Strategy for <i>C</i>-Glycosyl Bicyclo[1.1.1]pentanes. [PDF]
Qi C, Dell'Amico L, Goti G.
europepmc +1 more source
Total synthesis of asperdinones B, C, D, E and terezine D. [PDF]
Devarajappa R, Hanessian S.
europepmc +1 more source

