Results 251 to 260 of about 3,750,504 (279)

IP562083 a novel mGluR7 negative allosteric modulator

Pharmacological Reports, 2015
Piotr Brański, Grzegorz Burnat, Anna Stankiewicz, Ryszard Bugno, Maria Paluchowska, Katarzyna Kaczorowska, Barbara Chruścicka, Andrzej Bojarski, Andrzej Pilc   +8 more
openaire   +1 more source

Positive and negative allosteric modulation of GluK2 kainate receptors by BPAM344 and antiepileptic perampanel

Cell Reports, 2023
Alexander I Sobolevsky, Maria V. Yelshanskaya, Shanti P Gangwar   +2 more
exaly  

Small Molecules as Negative Allosteric Modulators of Alpha7 nAChRs

2012
VCU Theses and ...
openaire   +1 more source

The Negative Allosteric Modulator EU1794-4 Reduces Single-Channel Conductance and Ca2+ Permeability of GluN1/GluN2A N-Methyl-d-Aspartate Receptors

Molecular Pharmacology, 2021
Stephen C. Pelly, Riley E Perszyk, Stephen Traynelis   +2 more
exaly  

β-Arrestin-Biased Allosteric Modulator of NTSR1 Selectively Attenuates Addictive Behaviors

Cell, 2020
Alexandra Badea, Li Zibo, William C Wetsel   +2 more
exaly  

Identification of dual role of piperazine-linked phenyl cyclopropyl methanone as positive allosteric modulator of 5-HT and negative allosteric modulator of 5-HT receptors

European Journal of Medicinal Chemistry, 2019
Mohammad Imran Siddiqi, Prem N Yadav, Ajeet Kumar   +2 more
exaly  

Computer-aided design of negative allosteric modulators of NMDA receptor

Doklady Biochemistry and Biophysics, 2013
E V, Radchenko, D S, Karlov, A N, Zefirov, V A, Palyulin, N S, Zefirov, V M, Pentkovski   +5 more
openaire   +2 more sources

Discovery of VU0409106: A negative allosteric modulator of mGlu with activity in a mouse model of anxiety

Bioorganic and Medicinal Chemistry Letters, 2013
Kyle A. Emmitte, Craig W. Lindsley, Jeffrey Conn   +2 more
exaly  

DSR-98776, a novel selective mGlu receptor negative allosteric modulator with potent antidepressant and antimanic activity

European Journal of Pharmacology, 2015
Taro Kato
exaly  

ARYLSULFONAMIDE DERIVATIVES AS MGLUR4 NEGATIVE ALLOSTERIC MODULATORS

2021
BIEMANS BARBARA, GOBBI LUCA, JAESCHKE GEORG, KNUST HENNER, LINDEMANN LOTHAR, O'HARA FIONN, PLANCHER JEAN-MARC   +6 more
openaire   +2 more sources