In vitro toxicity of piperazine derivatives involves mitochondrial dysfunction and microtubule-related changes in neuronal cell models. [PDF]
BMC Pharmacol ToxicolRönnberg D, Jacobsson SOP.
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Design, Synthesis, and Biological Evaluation of Novel Dithiocarbamate-Based Human Carbonic Anhydrase IX/XII Inhibitors as Potential Anti-Glioblastoma Agents. [PDF]
MoleculesAltıntop MD +8 more
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Design and Synthesis of Novel Imidazo[4,5-c]pyridine Derivatives, Evaluation of Their Activity Against Hepatitis C Virus and In Silico Prediction of Their Binding Mode to NS4B Protein. [PDF]
ChemMedChemKarampella E +10 more
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Piperazine linked chitosan schiff base nanoparticles as a novel antibiofilm and antibacterial strategy against clinically relevant pathogens. [PDF]
Sci RepSoliman MM +6 more
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Structure-activity profiling of indazole-based derivatives as spinster homolog 2 (Spns2)-dependent S1P release inhibitors. [PDF]
Bioorg Med Chem LettHernandez M +7 more
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Targeting DYRK1A with rationally designed pyrazine-guanidine hybrids for Alzheimer's disease: design, synthesis, and biological evaluation. [PDF]
RSC AdvKhan S +9 more
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Structure-Affinity Relationship Optimization of SYA16263 Yields New Ligands with Improved Receptor Affinity and Antipsychotic-Like Properties. [PDF]
ACS OmegaGonela UM +9 more
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Prioritization of chemical scaffolds using the TDR Targets database: An integrative workflow for Trypanosoma cruzi drug discovery. [PDF]
PLoS Negl Trop DisUrán Landaburu L +3 more
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Noncovalent SARS-CoV-2 main protease inhibitors targeting the catalytic dyad and primed substrate binding subsites. [PDF]
RSC Med ChemBhandari D +9 more
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