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4-aminoquinolone piperidine amides: noncovalent inhibitors of DprE1 with long residence time and potent antimycobacterial activity.
Journal of Medicinal Chemistry, 2014 M. Naik, Vaishali Humnabadkar, S. Tantry, Manoranjan Panda, A. Narayan, S. Guptha, Vijender Panduga, P. Manjrekar, L. K. Jena, K. Koushik, Gajanan S Shanbhag, Sandesh Jatheendranath, M. Manjunatha, Gopinath Gorai, Chandramohan Bathula, Suresh S Rudrapatna, V. Achar, Sreevalli Sharma, Anisha Ambady, Naina Hegde, Jyothi Mahadevaswamy, P. Kaur, V. Sambandamurthy, Disha Awasthy, Chandan Narayan, S. Ravishankar, P. Madhavapeddi, J. Reddy, K. Prabhakar, R. Saralaya, M. Chatterji, James D. Whiteaker, Bob Mclaughlin, L. Chiarelli, G. Riccardi, M. Pasca, C. Binda, J. Neres, N. Dhar, Francois Signorino-Gelo, J. Mckinney, V. Ramachandran, R. Shandil, R. Tommasi, P. Iyer, S. Narayanan, V. Hosagrahara, Stefan L Kavanagh, Neela Dinesh, S. Ghorpade +49 moresemanticscholar +1 more source