Raltegravir: first in class HIV integrase inhibitor
Zelalem Temesgen1, Dawd S Siraj21Mayo Clinic, Rochester, MN, USA; 2East Carolina University Greenville, NC, USAAbstract: On October 16, 2007, the US Food and Drug Administration (FDA) approved raltegravir for treatment of human immunodeficiency virus ...
Zelalem Temesgen, Dawd S Siraj
doaj
Subgroup and Resistance Analyses of Raltegravir for Resistant HIV-1 Infection [PDF]
David A. Cooper+28 more
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Long-term efficacy and safety of raltegravir in the management of HIV infection
Michelle D Liedtke, C Ryan Tomlin, Staci M Lockhart, Misty M Miller, R Chris Rathbun Department of Clinical and Administrative Sciences, College of Pharmacy, University of Oklahoma Health Sciences Center, Oklahoma City, OK, USA Abstract: Raltegravir is ...
Liedtke MD+4 more
doaj
Raltegravir for HIV-1 infected children and adolescents: efficacy, safety, and pharmacokinetics
Kajal B Larson, Jennifer R King, Edward P Acosta Department of Pharmacology and Toxicology, University of Alabama at Birmingham, Birmingham, AL, USA Abstract: Raltegravir was the first HIV integrase strand-transfer inhibitor to be approved by the US FDA,
Larson KB, King JR, Acosta EP
doaj
Comparison of Raltegravir and Elvitegravir on HIV-1 Integrase Catalytic Reactions and on a Series of Drug-Resistant Integrase Mutants [PDF]
Jessica Marinello+5 more
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Switch from enfuvirtide (ENF) to raltegravir (RAL): a simplification option for heavily pretreated HIV patients (pts) [PDF]
Francesca Gatti+5 more
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AIM. To evaluate the efficiency and safety of using raltegravir (RAL) twice daily in conjunction with a once-daily fixed dose combination of abacavir (ABC)/lamivudine (3TC) in patients with HIV infection and active tuberculosis who have not previously ...
A V Kravchenko+7 more
doaj
No Residual Activity of Raltegravir After Development of 148 Complex Mutations In Vivo [PDF]
Homayoon Khanlou+2 more
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Effect of Tipranavir-Ritonavir on Pharmacokinetics of Raltegravir [PDF]
William D. Hanley+9 more
openalex +1 more source
Raltegravir, elvitegravir, and metoogravir: the birth of "me-too" HIV-1 integrase inhibitors [PDF]
Erik Serrao+3 more
openalex +1 more source