Results 31 to 40 of about 309 (104)

Pharmacological blockage of the AHR-CYP1A1 axis: a call for in vivo evidence. [PDF]

J Mol Med (Berl), 2022
Coelho NR, Pimpão AB, Correia MJ, Rodrigues TC, Monteiro EC, Morello J, Pereira SA.   +6 more
europepmc   +1 more source

Functional coupling of ATP-binding cassette transporter Abcb6 to cytochrome P450 expression and activity in liver. [PDF]

J Biol Chem, 2015
Chavan H, Li F, Tessman R, Mickey K, Dorko K, Schmitt T, Kumer S, Gunewardena S, Gaikwad N, Krishnamurthy P.   +9 more
europepmc   +1 more source

Synthesis, Characterization, and Biological Evaluation of Some Novel Pyrazolo[5,1-b]thiazole Derivatives as Potential Antimicrobial and Anticancer Agents. [PDF]

Molecules, 2021
Alsayari A, Muhsinah AB, Asiri YI, Al-Aizari FA, Kheder NA, Almarhoon ZM, Ghabbour HA, Mabkhot YN.   +7 more
europepmc   +1 more source

Wedelolactone, a natural coumestan with multiple pharmacological effects. [PDF]

Front Pharmacol
Han S, Li M, Yang L, Zhuang X.
europepmc   +1 more source

Synthesis, characterization and biological studies of pyrazole-linked Schiff bases and their copper(ii) complexes as potential therapeutics. [PDF]

RSC Adv
Kumari P, Kumar A, Kataria R, Kaushik NK, Ahmed M, Ansari A, Ekta, Brahma M, Maruthi M, Babu YS, Singh B, Kumar V.   +11 more
europepmc   +1 more source

Novel Regioselective Synthesis of 1,3,4,5-Tetrasubstituted Pyrazoles and Biochemical Valuation on F₁F_O-ATPase and Mitochondrial Permeability Transition Pore Formation. [PDF]

Pharmaceutics, 2023
Algieri V, Algieri C, Costanzo P, Fiorani G, Jiritano A, Olivito F, Tallarida MA, Trombetti F, Maiuolo L, De Nino A, Nesci S.   +10 more
europepmc   +1 more source

High-throughput, high-content screening for novel pigmentation regulators using a keratinocyte/melanocyte co-culture system. [PDF]

Exp Dermatol, 2014
Lee JH, Chen H, Kolev V, Aull KH, Jung I, Wang J, Miyamoto S, Hosoi J, Mandinova A, Fisher DE.   +9 more
europepmc   +1 more source

Design, synthesis, characterization, pharmacological evaluation and in silico ADMET and molecular docking and dynamics simulations of a novel series of N-substituted pyrazole from chalcone derivatives. [PDF]

Sci Rep
Hafez HN, Otaif HY, Alshammari BH, Alhebshe NS, El-Sayed AF, Abbas HS, Ammar RA.   +6 more
europepmc   +1 more source

An efficient eco-friendly, simple, and green synthesis of some new spiro-N-(4-sulfamoyl-phenyl)-1,3,4-thiadiazole-2-carboxamide derivatives as potential inhibitors of SARS-CoV-2 proteases: drug-likeness, pharmacophore, molecular docking, and DFT exploration. [PDF]

Mol Divers
El-Saghier AM, Enaili SS, Abdou A, Kadry AM.   +3 more
europepmc   +1 more source

Benzoxazole Derivative K313 Induces Cell Cycle Arrest, Apoptosis and Autophagy Blockage and Suppresses mTOR/p70S6K Pathway in Nalm-6 and Daudi Cells. [PDF]

Molecules, 2020
Zhong W, Tang X, Liu Y, Zhou C, Liu P, Li E, Zhong P, Lv H, Zou Q, Wang M.   +9 more
europepmc   +1 more source