Results 41 to 50 of about 1,134 (75)

6-Amino-4-phenylpyrrolo[2,3-c][1,2,6]thiadiazine-5-carbonitrile

open access: yes
The reaction of 2-(3-chloro-5-phenyl-4H-1,2,6-thiadiazin-4-ylidene)malononitrile with ammonia in anhydrous THF, at ca. 20 °C, for 24 h, gave 6-amino-4-phenylpyrrolo[2,3-c][1,2,6]thiadiazine-5-carbonitrile in 95% yield.
Panayiotis A. Koutentis   +2 more
core   +1 more source

1,2,6-Thiadiazinones as Novel Narrow Spectrum Calcium/Calmodulin-Dependent Protein Kinase Kinase 2 (CaMKK2) Inhibitors. [PDF]

open access: yesMolecules, 2018
Asquith CRM   +11 more
europepmc   +1 more source

Looking for Novel Capsid Protein Multimerization Inhibitors of Feline Immunodeficiency Virus. [PDF]

open access: yesPharmaceuticals (Basel), 2018
Sierra N   +5 more
europepmc   +1 more source

Postoperative analgesia by D-myo-inositol-1,2,6-trisphosphate in patients undergoing cholecystectomy

open access: yes, 1998
D-myo-inositol-1,2,6-trisphosphate (1,2,6-IP3) possesses antiinflammatory properties, such as reduced eicosanoid synthesis and inhibition of inflammation-induced edema. These properties suggest possible analgesic effects.
Cassuto, Jean,   +4 more
core  

Dibenzo[1,2,5]thiadiazepines are non-competitive GABAA receptor antagonists. [PDF]

open access: yesMolecules, 2013
Ramírez-Martínez JF   +8 more
europepmc   +1 more source

Topical D-myo-inositol-1,2,6-trisphosphate and hexylbetaine treatment reduces albumin extravasation in experimental rat skin burn injury

open access: yes, 1998
The anti-inflammatory agent D-myo-inositol-1,2,6-trisphosphate (1,2,6-IP3) has shown beneficial effects in experimental burns following systemic administration.
Cassuto, Jean,   +4 more
core  

Correction to "The Photochemical Mediated Ring Contraction of 4<i>H</i>-1,2,6-Thiadiazines To Afford 1,2,5-Thiadiazol-3(2<i>H</i>)-one 1-Oxides". [PDF]

open access: yesOrg Lett
Broumidis E   +12 more
europepmc   +1 more source

Synthesis of 1,2,6-Thiadiazin 1,1-Dioxide Derivatives as Trypanocidal Agents

open access: yes, 2014
: It describes the synthesis of new 1,2,6-Thiadiazin 1,1-dioxide derivatives using condensation of the Knoevenagel type.
A. Gómez-barrio   +5 more
core  

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