Selective Cycloaddition Reactions of Sulfo-Biginelli Derived 1,2,6-Thiadiazines
Modified sulfo-Biginelli conditions were developed to access dihydro-1,2,6-thiadiazines that were further functionalized and oxidized to 1,2,6-thiadiazines. These electron-deficient heterocyclic building blocks were subjected to regio- and stereoselective [4+2] and [3+2] cycloadditions with an electron-rich methylene cyclopropane, non-stabilized ...
Clare Hill, Michael Sambor, Peter Wipf
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