Results 71 to 80 of about 202 (136)

Stefano Marcaccini: a pioneer in isocyanide chemistry. [PDF]

open access: yesMol Divers
Neo AG   +4 more
europepmc   +1 more source

A Convenient One-Pot Synthesis of Novel Benzimidazole-Thiazinone Derivatives and Their Antimicrobial Activity. [PDF]

open access: yesAntibiotics (Basel)
Samreen S   +8 more
europepmc   +1 more source
Some of the next articles are maybe not open access.

Related searches:

Recent Advances in Synthesis and Medicinal Evaluation of 1,2‐Benzothiazine Analogues

Asian Journal of Organic Chemistry, 2022
AbstractBenzothiazines are one of the significant nitrogen containing heterocyclic scaffolds which are found to be multipurpose in the fields of drug discovery and medicinal chemistry. They are realized to be effective in curing enzymatic diseases caused by COX‐2, ALR‐2 (Aldose reductase enzyme), ALP (Alkaline phosphatase), 11β‐HSD 1 (11β ...
Reetu Reetu   +2 more
openaire   +1 more source

Regioselective Syntheses of 1,2‐Benzothiazines by Rhodium‐Catalyzed Annulation Reactions

Angewandte Chemie, 2015
AbstractRhodium‐catalyzed directed carbene insertions into aromatic CH bonds of S‐aryl sulfoximines lead to intermediates, which upon dehydration provide 1,2‐benzothiazines in excellent yields. The domino‐type process is regioselective and shows a high functional‐group tolerance. It is scalable, and the only by‐products are dinitrogen and water. Three
Ying, Cheng, Carsten, Bolm
openaire   +2 more sources

Synthesis and analgesic and anti-inflammatory activities of 1,2-benzothiazine derivatives

Archives of Pharmacal Research, 1999
Three 1,2-benzothiazine derivatives were synthesized, and their analgesic/anti-inflammatory efficacy and their effects on gastric irritation were evaluated. Among the three compounds, 39 exhibited the most potent analgesic action, but the effect was weaker than that of piroxicam.
E B, Lee, S K, Kwon, S G, Kim
openaire   +2 more sources

Rhodium-Catalyzed Oxidative Annulation of Sulfoximines and Alkynes as an Approach to 1,2-Benzothiazines

Angewandte Chemie - International Edition, 2013
Revitalization by oxygen: A rhodium(III)-catalyzed oxidative CH/NH activation/annulation sequence provided access to a variety of substituted 1,2-benzothiazine derivatives from readily available NH-sulfoximines and alkynes (see scheme; Cp*=C5 Me5 ). The oxidation system consisted of molecular oxygen in combination with a catalytic amount of Fe(OAc)2 .
Carsten Bolm   +2 more
exaly   +3 more sources

Multilevel topological description of molecular packings in 1,2-benzothiazines

CrystEngComm, 2014
A new method for description of molecular networks and packings is proposed and implemented into the program package TOPOS.
Farhana Aman   +6 more
openaire   +1 more source

Home - About - Disclaimer - Privacy