Results 171 to 180 of about 12,853,470 (222)

New 5-(pyridin-3-yl)-1,3,4-oxadiazoles derivatives as VEGFR2 inhibitors: <i>in silico</i> study, synthesis, and cytotoxicity evaluation. [PDF]

Res Pharm Sci
Abdulhussein AN, Oleiwi MA.
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Benzo[<i>d</i>]imidazole anchored oxadiazole derivatives: synthesis, characterization, biological evaluation, <i>in silico</i> docking and ADME-T analysis. [PDF]

RSC Adv
Salluri YR, Chepuri K, Anwar S.
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A Lactone-Enabled Approach to Metronidazole-Based Scaffolds. [PDF]

J Org Chem
Yu X, González-Montiel GA, Shit P, Chang M, Wiest O, Mobashery S.   +5 more
europepmc   +1 more source

Synthesis of Benzazolyl Oxadiazolyl/Thiadiazolyl/Triazolyl Amines and Their Antimicrobial, Antioxidant, In Silico and In Vivo Anti-Inflammatory Activities. [PDF]

Chem Biodivers
Madduru K, Donthamsetty VS, Begum S, Venkatapuram P.   +3 more
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Sulfonamide-Based 2-Amino-1,3,4-Oxadiazole Derivatives as Dual Cholinesterase and Carbonic Anhydrase Inhibitors: Design, Synthesis, Kinetic Characterization, Molecular Modeling, and ADMET Evaluation. [PDF]

Drug Dev Res
Arslan Karahan G, Gökçe B, Muhammed MT, Ayan EK, Özçelik AB.   +4 more
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Experimental and MEDT Study of Sydnone-Alkyne Cycloaddition-Based Synthesis of 1,4-Disubstituted Pyrazoles and In Silico Investigation of Their Binding to HCV and HIV Proteins. [PDF]

Molecules
Zerbib S, Eddahmi M, Alaqarbeh M, Bodet PE, Thiery V, Fatimi A, Cruz-Martins N, Bailly C, Domingo LR, Bouissane L.   +9 more
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Rational design of naphtho[2,3-<i>d</i>]imidazole-4,9-dione-linked 1,3,4-oxadiazoles as α-amylase inhibitors supported by QSAR, docking, molecular dynamics, and ADME approaches. [PDF]

RSC Adv
Devi M, Kumar P, Singh R, Sindhu J, Kumar A, Lal S, Singh D, Kumar H.   +7 more
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Structural Modifications of Nonsteroidal Anti-Inflammatory Drugs (NSAIDs): New Horizons in Antimicrobial Drug Discovery. [PDF]

Arch Pharm (Weinheim)
Koçak Aslan E, Karagüzel A, Gündüz MG.   +2 more
europepmc   +1 more source

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A OVERVIEW ON ANTIMICROBIAL AND ANTI-INFLAMMATORY ACTIVITY OF 1, 3, 4-OXADIAZOLES

INDIAN DRUGS, 2020
1, 3, 4-oxadiazoles first came into the lime light about 80 years ago. With the increasing world population, the number of microbial infections has increased all over. To overcome the continuously spreading harmful microbial infections, the need for newer and newer drugs has increased tremendously.
Satvir Singh, Manpreet Kaur, Divya Bhandari, Mandeep Kaur, Monika Gupta   +4 more
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1, 2, 4-Oxadiazoles

1976
Publisher Summary This chapter focuses on the chemistry of 1,2,4-oxadiazoles and the corresponding reduced derivatives. The chapter discusses the synthesis of 1,2,4-oxadiazoles. Two widely used general methods of synthesizing 1,2,4-oxadiazoles embrace 95% of the practical preparations of these compounds: The conversion of amidoximes by means of ...
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