Results 151 to 160 of about 3,911 (190)

Acid Versus Amide-Facts and Fallacies: A Case Study in Glycomimetic Ligand Design. [PDF]

Molecules
Smieško M, Jakob RP, Mühlethaler T, Preston RC, Maier T, Ernst B.   +5 more
europepmc   +1 more source

Stereochemical Analysis of Tertiary Trifluoroacetamides Leveraging Both Through-Space ¹H···¹⁹F Spin-Spin Couplings and Anisotropic Solvent-Induced Shifts. [PDF]

J Org Chem
Watanabe K, Takano R, Tabata H, Hirano K, Iida M, Oshitari T, Natsugari H, Kusumi T, Nakamura K, Takahashi H.   +9 more
europepmc   +1 more source

Ultrasonic-assisted, additive-free Pd-catalyzed Suzuki-Miyaura cross-coupling enabled synthesis of novel arylated benzofuran-triazole hybrids. [PDF]

Front Chem
Saif MJ, Ahmad S, Mushtaq A, Munawar S, Zahoor AF, Ettampola S, Irfan A, Kotwica-Mojzych K, Ruszel K, Mojzych M.   +9 more
europepmc   +1 more source

Solvent-controlled, chemodivergent oxidative anionic Fries rearrangement of <i>O</i>-aryl carbamates under aerobic conditions. [PDF]

Chem Sci
Gnavi R, De Nardi F, Meazzo C, Ghinato S, Grimaldi E, Maranzana A, Prandi C, Blangetti M.   +7 more
europepmc   +1 more source

Discovery and Characterization of Divarasib (GDC-6036), a Potent Covalent Inhibitor of KRAS G12C. [PDF]

J Med Chem
Endres NF, Do S, Mroue R, Terrett JA, Saabye M, Oh A, Hunsaker T, Chan E, Tran JC, Nguyen LK, Lian Q, Ma TP, Garner T, Gerosa L, Beresini M, Boudreau A, Bronner SM, Cyr P, Ishisoko N, Izrayelit Y, Jiang F, Kellar T, La H, Labadie S, Lardy M, Liu L, Liu W, Miller S, Rudolph J, Plise E, Sellers BD, Shao C, Wang W, Wang Y, Wei W, Wong S, Yu C, Yu K, Yuen PW, Zang R, Zhang C, Zhou Y, Zhu X, Quinn JG, Ye X, Kiefer JR, Mao J, Evangelista M, Merchant M, Landry ML, Malhotra S, Purkey HE.   +51 more
europepmc   +1 more source

Synthesis and evaluation of quinolinvinyl-phenoxy-1,2,3-triazole-acetamide hybrids against breast cancer. [PDF]

Sci Rep
Safavi M, Iraji A, Farid SM, Mahdavi M, Fattaheian-Dehkordi S, Akbarzadeh T, Saeedi M.   +6 more
europepmc   +1 more source

Resistance Analysis of Low-Level Virologic Rebound During HIV-1 Treatment With Lenacapavir and Broadly Neutralizing Antibodies Teropavimab and Zinlirvimab. [PDF]

J Infect Dis
Selzer L, Demirdjian S, Falkard B, Li J, Martin R, Collins SE, Eron J, VanderVeen LA, Callebaut C.   +8 more
europepmc   +1 more source

Reprogramming Imine Reductases for Enantioselective Reduction of Electron-Rich Enamides. [PDF]

JACS Au
Liu XQ, Li R, Chen JL, Li Y, Wei L, Wu H, Li L, Chen BH, Wu Y, Liu SJ, Lin GX, Zhang JF, Zheng Y, Zhang C, Yang YF, Wang X, Chen P, Jia ZJ.   +17 more
europepmc   +1 more source

Investigation of Natural Resistance to Fostemsavir and Lenacapavir in Naïve Primary Infections by Ultra-Deep Sequencing of near Full-Length HIV-1 Genomes. [PDF]

Viruses
Lazzari E, Rozera G, Gagliardini R, Mazzotta V, Fabeni L, Forbici F, Berno G, Cosentino C, Girardi E, Antinori A, Maggi F, Abbate I.   +11 more
europepmc   +1 more source

Diastereoselective Cyclopropanation with Secondary Diazoacetamides to Access <i>endo</i>-Azabicyclo[3.1.0]hexane-6-carboxamides. [PDF]

Org Lett
Nguyen TH, Saito T, Chang W, Navarro A, Davies HML.   +4 more
europepmc   +1 more source