Results 141 to 150 of about 7,268 (257)

Fixed into acetamides [PDF]

Nature Catalysis, 2019
openaire   +1 more source

A Sustainable Borrowing Hydrogen Strategy in Natural Deep Eutectic Solvents for the N‐Alkylation of Amines From Alcohols

European Journal of Organic Chemistry, Volume 29, Issue 16, 25 April 2026.
A sustainable, ligand‐free Pd‐catalyzed borrowing hydrogen protocol in a biodegradable hydrophobic natural deep eutectic solvent (NADES) (thymol/DL‐menthol) enables the N‐alkylation of primary amines with benzylic alcohols under mild, aerobic conditions, allowing efficient reuse of both catalyst and solvent for seven consecutive cycles. The hydrophobic
Maryam Saeb, Maristella Simone, Luciana Cicco, Paola Vitale, Filippo Maria Perna, Vito Capriati   +5 more
wiley   +1 more source

Synthesis of Sulfur Heterocycles by Palladium‐Catalyzed Cyclization

European Journal of Organic Chemistry, Volume 29, Issue 14, 15 April 2026.
In spite of the well‐known palladium thiophilicity, sulfur‐containing acyclic substrates may efficiently undergo several different kinds of palladium‐catalyzed cyclization processes leading to highly important sulfur heterocycles in one synthetic step. Advances in this challenging and stimulating field of research are presented in this review.
Bartolo Gabriele
wiley   +1 more source

Identification of α-Azacyclic Acetamide-Based Inhibitors of <i>P. falciparum</i> Na⁺ Pump (<i>Pf</i>ATP4) with Fast-Killing Asexual Blood-Stage Antimalarial Activity by Phenotypic Screening. [PDF]

ACS Infect Dis
Casas A, Imlay LS, Thathy V, Fairhurst KJ, Lehane AM, Lawong AK, Deni I, Striepen J, Lee S, Kumar A, Xing C, Niederstrasser H, Posner BA, Laleu B, Charman SA, Fidock DA, Ready JM, Phillips MA.   +17 more
europepmc   +1 more source

EDA Complex–Mediated C(sp3)–H Cross‐Dehydrogenative Coupling Enables Synthesis of Noncanonical α,β‐Diamino Acids

European Journal of Organic Chemistry, Volume 29, Issue 14, 15 April 2026.
Access to nonproteinogenic α,β‐diamino acids from simple feedstock precursors is of great interest to generate medicinal small molecule libraries. We report a regioselective photoinduced C(sp3)–C(sp3) cross‐dehydrogenative coupling (CDC) of N‐arylglycine derivatives with amides.
Krishnakumar Sachidanandan, Cole Stenftenagel, Athul Joshy, Alexander M. Cluff, Sébastien Laulhé   +4 more
wiley   +1 more source

Radioiodination of Two Carborane‐Based Dual Cyclooxygenase‐2/5‐Lipoxygenase Inhibitors and Their In Vitro and In Vivo Evaluation

ChemBioChem, Volume 27, Issue 7, 14 April 2026.
Two dicarbadodecaborane(12)‐based dual cyclooxygenase‐2/5‐lipoxygenase (COX‐2/5‐LO) inhibitors were 123I‐labeled. Refinement of labeling and formulation conditions and extensive in vitro characterization are presented. Cell uptake studies in COX‐2‐ and 5‐LO‐overexpressing cell lines showed COX‐2‐independent and partly 5‐LO‐dependent uptake.
Jonas Schädlich, Martin Ullrich, Cathleen Haase‐Kohn, Robert Wodtke, Sebastian Braun, Maximilian Molitor, Bettina Hofmann, Dieter Steinhilber, Klaus Kopka, Evamarie Hey‐Hawkins, Jens Pietzsch, Markus Laube   +11 more
wiley   +1 more source

Synthesis of 2-(Quinoxalin-2-yl)acetamides and Their Preliminary Cytotoxic and Antibacterial Activity. [PDF]

Chem Biodivers
Tovar-Roman CE, Hernández-Vázquez E, Rivera-Chávez JA.   +2 more
europepmc   +1 more source

Pesticide Use in the 1983 Soybean Crop: Report of a Survey of Arkansas Producers [PDF]

, 1985
Waldrum, Joseph D.
core   +2 more sources

N-(Alkylsulfamoyl)aldimines: easily deprotected precursors for diarylmethylamine synthesis [PDF]

, 2013
Awano, Cao, Catt, Crampton, Dahmen, Duan, Iso, Jagt, Klinger, Luo, Marques, Martin Fox, Masui, Nachbaur, Oi, Okamoto, Otomaru, Pflum, Ramadhar, Rosemary H. Crampton, Sanz, Shintani, Simon Woodward, Tokunaga, Tsai, Ueda, Weix, Winum   +27 more
core   +2 more sources

The Multifaceted Legacy of Thalidomide: Chemistry and Biology Driving Modern Drug Design

ChemMedChem, Volume 21, Issue 7, 14 April 2026.
Thalidomide serves as a molecular nexus linking chemistry and biology: advances in synthesis and structural understanding enable protein degradation technologies, while its immunomodulatory activity underpins anti‐inflammatory and anticancer therapies.
Konstantina Nikovia, Michael Kapsalis, Michael Georgoulakis, Athanasios Panousis, Constantinos G. Neochoritis   +4 more
wiley   +1 more source