Results 31 to 40 of about 7,268 (257)

The search for the 'next' euphoric non-fentanil novel synthetic opioids on the illicit drugs market: current status and horizon scanning [PDF]

, 2019
Purpose: A detailed review on the chemistry and pharmacology of non-fentanil novel synthetic opioid receptor agonists, particularly N-substituted benzamides and acetamides (known colloquially as U-drugs) and 4-aminocyclohexanols, developed at the Upjohn ...
A Helander, A Regina La, A Schneir, AG Hayes, AG Hayes, AJ Krotulski, AJ Krotulski, ALA Mohr, C McKenzie, C Soussan, Craig McKenzie, D Fabregat-Safont, D Lednicer, D Lednicer, D Lednicer, D Lednicer, D Lednicer, D Papsun, E Gerace, GW Peng, I Metushi, IM McIntyre, J Seither, J Szmuszkovicz, J Szmuszkovicz, JB Zawilska, JK O’Donnell, K Domanski, K Koch, KA Rambaran, Kirti Kumari Sharma, KN Ellefsen, KT Vo, L Ventura, M Dziadosz, M Katselou, MC Hout Van, MH Baumann, MJ Jones, MP Prekupec, Niamh NicDaeid, NJ Harper, P Armenian, P Armenian, P Nikolaou, PF Voigtlander Von, PF Voigtlander Von, PF Voigtlander Von, RA Fujimoto, RA Lahti, RT Brittain, SA Harding, SC Ifeagwu, SP Elliott, Tim G. Hales, TP Rohrig, USAN Council, V Coopman, Vaidya Jayathirtha Rao, W Fleming, X Ruan, Z Davey, Z Li, ZH Liu   +63 more
core   +2 more sources

Direct acylation of aryl amines using dimethylformamide and dimethylacetamide as the acyl resources

Journal of Saudi Chemical Society, 2016
The treatment of aryl amines with dimethylformamide (DMF) and dimethylacetamide (DMA) in the presence of hydrochloric acid brings about efficient N-acylation to give the corresponding aryl formamides and aryl acetamides in acceptable to excellent yields.
Qing Zhang, Cui Chen
doaj   +1 more source

LXXXIII.—Mercury acetamide [PDF]

J. Chem. Soc., Trans., 1898
n ...
openaire   +1 more source

Spectroscopic and Theoretical Studies of Some 3-(4 '-Substituted phenylsulfanyl)-1-methyl-2-piperidones [PDF]

, 2013
The analysis of the IR carbonyl bands of some 3-(4 '-substituted phenylsulfanyl)1- methyl-2-piperidones 1-6 bearing substituents: NO2 (compound 1), Br (compound 2), Cl (compound 3), H (compound 4) Me (compound 5) and OMe (compound 6) supported by B3LYP ...
Bruna Contieri, Carlos R. Cerqueira, Daniel N. S. Rodrigues, Elisângela Vinhato, Jean M. M. Santos, Jr, Julio Zukerman-Schpector, Maurizio Dal Colle, Paulo R. Olivato   +8 more
core   +2 more sources

Synthesis, structure and properties of N-R-2-(5-(5-methyl-1H-pyrazole-3-yl)-4-phenyl-4H-1,2,4-triazole-3-ylthio)acetamides

Aktualʹnì Pitannâ Farmacevtičnoï ì Medičnoï Nauki ta Praktiki, 2019
Heterocyclic compounds remain the most promising group of compounds, through which the new drugs with characteristic list of properties are successfully created. Examples of this systems are 1,2,4-triazole and pyrazole.
A. S. Hotsulia, S. O. Fedotov
doaj   +1 more source

Coordination chemistry of amide-functionalised tetraazamacrocycles: structural, relaxometric and cytotoxicity studies [PDF]

, 2010
Three different tetraazamacrocyclic ligands containing four amide substituents that feature groups (namely allyl, styryl and propargyl groups) suitable for polymerisation have been synthesised.
Aime, Aime, Aime, Aime, Aime, Ali, Andrew J. P. White, Antoni, Beeta Balali-Mood, Behnam Azad, Bottrill, Bryson, Burdinski, Caravan, Cattaneo, Chapon, Cheng, Cilliers, De Leon-Rodriguez, De Leon-Rodriguez, Delgado, Faulkner, Fields, Gabriel, Guo, Hermann, Iten, Joachim H. G. Steinke, Jonathan Martinelli, Kaneshiro, Langereis, Major, Mani, Mark F. Lythgoe, Maumela, Montgomery, Moore, Muller, New, Oliver, Patrizia Ferretti, Pratesi, Rachael Panizzo, Ramon Vilar, Roosenburg, Schlesinger, Tan, Trokowski, Villaraza, Viola-Villegas, Viswanathan, Wu, Xu, Zhang, Zucchi   +54 more
core   +1 more source

Structural and Compositional Effects on the Scintillation Properties of Fast Emitting Metal‐Organic Frameworks

Advanced Science, EarlyView.
The crystalline structure, the atomic numbers of the constituent elementsand the size of MOF crystals each influence their photoluminescence and scintillation properties in distinct ways. Together, these factors provide valuable guidelines for designing systems with optimized performance and tunable timing characteristics, arising from the synergistic ...
Francesca Cova, Jacopo Perego, Biplab Joarder, Nobuhiro Yanai, Anna Vedda, Silvia Bracco, Angiolina Comotti, Angelo Monguzzi, Irene Villa   +8 more
wiley   +1 more source

Synthesis of Tetrahydroberberine N,N-Derived O-Acetamides

Molbank
The reaction of berberine derivatives containing at the O-9 position N,N-disubstituted acetamide fragments with sodium borohydride in methanol at 0 °C leads to a mild reduction of the “C” cycle with the formation of corresponding tetrahydroberberine ...
Ivan Vasil’evich Nechepurenko, Nina Ivanovna Komarova, Nariman Faridovich Salakhutdinov   +2 more
doaj   +1 more source

New thioxothiazolidinyl-acetamides derivatives as potent urease inhibitors: design, synthesis, in vitro inhibition, and molecular dynamic simulation

Scientific Reports, 2023
To identify potent urease inhibitors, in the current study, a series of thioxothiazolidinyl-acetamides were designed and synthesized. The prepared compounds were characterized by spectroscopic techniques, including FTIR, 1HNMR, 13CNMR, and elemental ...
Navid Dastyafteh, Milad Noori, Mohammad Nazari Montazer, Kamiar Zomorodian, Somayeh Yazdanpanah, Aida Iraji, Minoo Khalili Ghomi, Shahrzad Javanshir, Mehdi Asadi, Mehdi Dianatpour, Mahmood Biglar, Bagher Larijani, Massoud Amanlou, Mohammad Mahdavi   +13 more
doaj   +1 more source

Expanding the palette of phenanthridinium cations [PDF]

, 2014
5,6-Disubstituted phenanthridinium cations have a range of redox, fluorescence and biological properties. Some properties rely on phenanthridiniums intercalating into DNA, but the use of these cations as exomarkers for the reactive oxygen species (ROS ...
Acevedo, Amann, Amatore, Amii, Augustine, Barluenga, Blanchot, Blanksby, Bolognesi, Bourne, Bourne, Bourne, Chen, Cheng, Chiavarino, Chiavarino, Chéron, Coe, Darzynkiewicz, Deb, Diaba, Dimiza, Döbele, Exner, Fernández, García, Ghaneolhosseini, Giroldo, Glendening, Glendening, Glendening, Glukhovtsev, Goerigk, Goryunov, Hata, Hu, Huang, Huber, Ihmels, Intrieri, Ishihara, Ishii, Jain, Jankowiak, Jones, Jose, Kitson, Korotvicka, Kostiainen, Kubar, Kundu, Lallana, Lee, Leupin, Lewis, Liang, Liljenberg, Liljenberg, Liljenberg, Liu, Liu, Logan, Luedtke, Luedtke, Manetsch, Marivingt-Mounir, Marivingt-Mounir, Mayer, McBurney, Michalski, Michels, Molander, Nakanishi, O′Brien, O′Connor, Parenty, Park, Pliego, Prunkl, Radic, Rangarajan, Richmond, Robinson, Schmidt, Shaw, Sletten, Smith, Sotomayor, Stevens, Stojkovic, Sumerlin, Sun, Suzuki, Takeda, Tanaka, Tanaka, Tobisu, van der Wiel, Veale, Wainwright, Wakelin, Walls, Watkins, Weigend, Weinhold, Weinhold, Wolff, Yamaguchi, Zhang, Zhao, Zhao, Zhidkov, Zhidkov, Zielonka, Zille   +114 more
core   +4 more sources