Results 141 to 150 of about 1,971,711 (246)

Angiotensin I–Converting Enzyme Inhibitors Are Allosteric Enhancers of Kinin B1 and B2 Receptor Function [PDF]

, 2010
Ervin G. Erdös, Fulong Tan, Randal A. Skidgel   +2 more
openalex   +1 more source

Transplanting allosteric control of enzyme activity by protein–protein interactions: Coupling a regulatory site to the conserved catalytic core

, 2002
Aaron C. Pawlyk, Donald W. Pettigrew
openalex   +1 more source

Tailor-Made Enzyme Carriers: Preparation and Use of Adsorbents Specifically Designed to Immobilize Allosteric Enzymes in Activated Conformation [PDF]

, 2010
Salemi
openalex   +1 more source

Small molecule-mediated allosteric activation of the base excision repair enzyme 8-oxoguanine DNA glycosylase and its impact on mitochondrial function [PDF]

, 2022
Gaochao Tian, Steven R. Katchur, Yong Jiang, Jacques Briand, Michael D. Schaber, Constantine Kreatsoulas, Benjamin J. Schwartz, Sara H. Thrall, Alicia Davis, Sam Duvall, Brett A. Kaufman, William L. Rumsey   +11 more
openalex   +1 more source

BMS-345541 Is a Highly Selective Inhibitor of IκB Kinase That Binds at an Allosteric Site of the Enzyme and Blocks NF-κB-dependent Transcription in Mice

, 2003
James R. Burke, Mark A. Pattoli, Kurt R. Gregor, Patrick Brassil, John F. MacMaster, Kim W. McIntyre, Xiaoxia Yang, Violetta S. Iotzova, Wendy Clarke, Joann Strnad, Yuping Qiu, F. Christopher Zusi   +11 more
openalex   +1 more source

Single Enzyme Studies Reveal the Existence of Discrete Functional States for Monomeric Enzymes and How They Are “Selected” upon Allosteric Regulation [PDF]

, 2012
Nikos S. Hatzakis, Li W, Sune K. Jørgensen, Andreas H. Kunding, Pierre‐Yves Bolinger, Nicky Ehrlich, Ivan Makarov, Michael Skjøt, Allan Svendsen, Per Hedegård, Dimitrios Stamou   +10 more
openalex   +1 more source

Designing Allosteric Control into Enzymes by Chemical Rescue of Structure [PDF]

, 2012
Katelyn Deckert, S. Jimmy Budiardjo, Luke C. Brunner, Scott Lovell, John Karanicolas   +4 more
openalex   +1 more source

Discovery of novel allosteric inhibitors of HCV NS3/4a enzyme via structure-based drug design [PDF]

, 2012
Puja Pathuri, S. Saalau-Bethell, Andrew Woodhead, Maria G. Carr, Gianni Chessari, Joe Coyle, Martyn Frederickson, Brent Graham, C. Hamlett, S. Hiscock, Finn P. Holding, Harren Jhoti, Rachel McMenamin, Christopher W. Murray, Michael Reader, David C. Rees, Sharna J. Rich, Caroline J. Richardson, N. Thompson, Marcel L. Verdonk, M. Vinković, Paul A. Williams, Jeannine M. Yon   +22 more
openalex   +1 more source

Uncovering the Role of Distal Regions in PDK1 Allosteric Activation. [PDF]

ACS Bio Med Chem Au
Mulpuri N, Yao XQ, Hamelberg D.
europepmc   +1 more source

Decoding allosteric landscapes: computational methodologies for enzyme modulation and drug discovery. [PDF]

RSC Chem Biol
Zhu R, Wu C, Zha J, Lu S, Zhang J.
europepmc   +1 more source