Results 81 to 90 of about 36,012 (161)

Allosteric modulation and biased signalling at free fatty acid receptor 2. [PDF]

Nature
Zhang X, Guseinov AA, Jenkins L, Valentini A, Marsango S, Schultz-Knudsen K, Ulven T, Rexen Ulven E, Tikhonova IG, Milligan G, Zhang C.   +10 more
europepmc   +1 more source

Allosteric Modulation of Cannabinoid Type 1 Receptor by ZCZ011: Integration of In Vitro Pharmacology and Molecular Dynamics Simulation. [PDF]

ACS Bio Med Chem Au
Yadav TC, Swaminathan LI, Chirasani VR, Wu Z, Lu D, Ignatowska-Jankowska BM, Lichtman AH, Fitting S, Yadav-Samudrala BJ.   +8 more
europepmc   +1 more source

Efficient Characterization of GPCRs Allosteric Modulation: Application to the Rational Design of De Novo S1PR1 Allosteric Modulators. [PDF]

J Chem Inf Model
Cruz A, Warshel A.
europepmc   +1 more source

GluN2B-specific NMDAR positive allosteric modulation reverses cognitive and behavioral abnormalities in <i>Mecp2</i> and <i>Disc1</i> transgenic mice. [PDF]

Sci Adv
Ge Y, Tian T, Li B, Axerio-Cillies P, Chen W, Qin X, Zhao M, Sun QC, Li J, Floresco SB, Liu L, Yang X, Wang YT.   +12 more
europepmc   +1 more source

Long-Range Allosteric Modulation of DNA Duplex Dynamics Induced by Pyrrole-Imidazole Polyamide Binding. [PDF]

J Phys Chem Lett
Kendall-Price SET, Nichol RJO, Taladriz-Sender A, Phelps R, Malakar P, Greetham GM, Burley GA, Hunt NT.   +7 more
europepmc   +1 more source

Negative Allosteric Modulation of Agonist-Induced M₂ Muscarinic Receptor/β-Arrestin Interaction by Serum Autoantibodies from Patients with Chronic Chagas Disease. [PDF]

Cells
Carrera Páez LC, Beltrame SP, Auger SR, Sabra AH, Bilder CR, Irurzun IM, Waldner CI, Goin JC.   +7 more
europepmc   +1 more source

Allosteric modulation and direct activation of glycine receptors by a tricyclic sulfonamide. [PDF]

Sci Rep
Lara CO, Burgos CF, Fariña-Oliva K, Marileo AM, Martín VPS, Flaig D, Soto-Ortega P, Contreras OV, Sazo A, Gaete-Riquelme K, Corradi J, Muñoz-Montesino C, Fuentealba J, Castro PA, Aguayo LG, Bouzat C, Moraga-Cid G, Yévenes GE.   +17 more
europepmc   +1 more source

Allosteric modulation of Plasmodium falciparum Isoleucyl tRNA synthetase by South African natural compounds. [PDF]

PLoS One
Chepsiror C, Veldman W, Olotu F, Tastan Bishop Ö.   +3 more
europepmc   +1 more source

Structural basis for allosteric modulation of M. tuberculosis proteasome core particle. [PDF]

Nat Commun
Turner M, Uday AB, Velyvis A, Rennella E, Zeytuni N, Vahidi S.   +5 more
europepmc   +1 more source

Unraveling GPCRs Allosteric Modulation. Cannabinoid 1 Receptor as a Case Study. [PDF]

Proteins
Cruz A, Warshel A.
europepmc   +1 more source