Results 71 to 80 of about 3,108,804 (226)

Development of a fluorogenic small substrate for dipeptidyl peptidase-4

Beilstein Journal of Organic Chemistry, 2017
A series of aniline and m-phenylenediamine derivatives with electron-withdrawing 3,3,3-trifluoropropenyl substituents were synthesized as small and chemically stable fluorescent organic compounds.
Futa Ogawa, Masanori Takeda, Kanae Miyanaga, Keita Tani, Ryuji Yamazawa, Kiyoshi Ito, Atsushi Tarui, Kazuyuki Sato, Masaaki Omote   +8 more
doaj   +1 more source

Hydrogen bonding in C-methylated nitroanilines : the three-dimensional framework structure of 2-methyl-4-nitroaniline [PDF]

, 2001
Peer reviewedPublisher ...
Ferguson, G, Glidewell, C, Low, J N, Skakle, Jan, Wardell, J L   +4 more
core   +1 more source

Aniline-Tetramic Acids from the Deep-Sea-Derived Fungus Cladosporium sphaerospermum L3P3 Cultured with the HDAC Inhibitor SAHA.

Journal of Natural Products, 2018
Four new tetramic acids, cladosins H-K (1-4), and a related known compound, cladodionen (5), were isolated from the culture of the Mariana Trench (depth 6562 m) sediment-derived fungus Cladosporium sphaerospermum L3P3 treated with the histone deacetylase
Zhenzhen Zhang, Xueqian He, Guangwei Wu, Congcong Liu, Changjun Lu, Q. Gu, Qian Che, T. Zhu, Guojian Zhang, Dehai Li   +9 more
semanticscholar   +1 more source

Scope and Mechanistic Study of the Ruthenium-Catalyzed \u3cem\u3eortho\u3c/em\u3e-C−H Bond Activation and Cyclization Reactions of Arylamines with Terminal Alkynes [PDF]

, 2005
The cationic ruthenium hydride complex [(PCy3)2(CO)(CH3CN)2RuH]+BF4- was found to be a highly effective catalyst for the C−H bond activation reaction of arylamines and terminal alkynes.
Yi, Chae S., Yun, Young
core   +1 more source

Structural optimization and biological evaluation of 2-substituted 5-hydroxyindole-3-carboxylates as potent inhibitors of human 5-lipoxygenase. [PDF]

, 2009
Pharmacological suppression of leukotriene biosynthesis by inhibitors of 5-lipoxygenase (5-LO) is a strategy to intervene with inflammatory and allergic disorders.
BÜHRING U, KARG EM, LUDERER S, NORTHOFF H, PERGOLA C, ROSSI, ANTONIETTA, SAUTEBIN, LIDIA, TROSCHÜTZ R, WERZ O.   +8 more
core   +1 more source

Removal of Phenol and Aniline from Aqueous Solutions by Using Adsorption on to Pistacia terebinthus: Study of Adsorption Isotherm and Kinetics

تحقیقات سلامت در جامعه, 2017
Introduction and purpose: Aniline and phenol are used in a wide range of industries, namely dye material, rubber, pesticide, plastic, and paint industries. These chemicals are released to the environment via effluent.
shahin ahmadi, somaye rahdar
doaj  

Design, Synthesis and Preliminary Pharmacological Evaluation of New Non-Steroidal Anti-Inflammatory Agents Having a 4-(Methylsulfonyl) Aniline Pharmacophore

Molecules, 2012
A series of 4-(methylsulfonyl)aniline derivatives were synthesized in order to obtain new compounds as a potential anti-inflammatory agents with expected selectivity against COX-2 enzyme. In vivo acute anti-inflammatory activity of the final compounds 11–
Akeel Abdul Kadhum Jassim, Mohamed Hassan Mohammed, Monther Faisel Mahdi   +2 more
doaj   +1 more source

Radiosynthesis, in vitro and preliminary in vivo evaluation of the novel glutamine derived PET tracers [18F]fluorophenylglutamine and [18F]fluorobiphenylglutamine

, 2020
INTRODUCTION: Glucose has been deemed the driving force of tumor growth for decades. However, research has shown that several tumors metabolically shift towards glutaminolysis.
Baguet, Tristan, Beyzavi, M. Hassan, De Lombaerde, Stef, De Vos, Filip, Descamps, Benedicte, Donche, Sam, Goethals, Ingeborg, Hu, Jiyun, Lambe, Patricia, Pauwelyn, Glenn, Piron, Sarah, Vanhove, Christian, Verhoeven, Jeroen   +12 more
core   +1 more source

Dyeing of Polyester and Nylon with Semi-synthetic Azo Dye by Chemical Modification of Natural Source Areca Nut

Natural Products and Bioprospecting, 2017
Various azo compounds (Modified dyes) have been synthesised by chemical modification of areca nut extract (epicatechin), a plant-based Polyphenolic compound to get semi-synthetic dyes.
Ashitosh B. Pawar, Sandeep P. More, R. V. Adivarekar   +2 more
doaj   +1 more source

Pot, atom and step economic (PASE) synthesis of highly functionalized piperidines: a five-component condensation [PDF]

, 2007
The diastereoselective pot, atom and step economic (PASE) synthesis of highly functionalized piperidines has been realized. The procedure simply involves mixing methyl acetoacetate, 2 equiv of aldehyde and 2 equiv of aniline together in the presence of ...
Clarke, Paul A., Whitwood, Adrian C., Zaytzev, Andrey V.   +2 more
core   +1 more source