PBA2, a novel inhibitor of the β-catenin/CBP pathway, eradicates chronic myeloid leukemia including BCR-ABL T315I mutation. [PDF]
Yang K +8 more
europepmc +1 more source
In Silico Molecular Modeling of Four New Afatinib Derived Molecules Targeting the Inhibition of the Mutated Form of BCR-ABL T315I. [PDF]
Rocha KML +3 more
europepmc +1 more source
Correction for Kuroda et al., Bim and Bad mediate imatinib-induced killing of Bcr/Abl<sup>+</sup> leukemic cells, and resistance due to their loss is overcome by a BH3 mimetic. [PDF]
europepmc +1 more source
Rationally designed BCR-ABL kinase inhibitors for improved leukemia treatment via covalent and pro-/dual-drug targeting strategies. [PDF]
Sun J +11 more
europepmc +1 more source
The clinical significance of TAT, PIC, TM, and t-PAIC in vascular events of BCR/ABL-negative myeloproliferative neoplasms. [PDF]
Huang K +6 more
europepmc +1 more source
Molecular Modeling of Single- and Double-Hydrocarbon-Stapled Coiled-Coil Inhibitors against Bcr-Abl: Toward a Treatment Strategy for CML. [PDF]
Lima MCP +3 more
europepmc +1 more source
Concomitant L248V With E225V Mutation in the BCR-ABL Gene Associated With Rapid Chronic Myeloid Leukemia Lymphoid Blast Crisis. [PDF]
Tungjitviboonkun S +2 more
europepmc +1 more source

