Pitstop 2 binds to the clathrin terminal domain. This work explores the nature of the benzylidene moiety, R. The synthesis of 56 novel analogues reveals enhanced potency of a multiple analogues, with catechol‐free 2,3‐dihydroxybenzo[b][1,4]dioxone (54) returning a 1.2 μm IC50, ca 10‐fold more active than Pitstop 2. Pitstop 2, (Z)‐N‐(5‐(4‐bromenzylidene)
Kate Prichard+10 more
wiley +1 more source
Optimal photosynthesis of 2-benzothiazoles over hexaazatrinaphthylene-based porous aromatic frameworks. [PDF]
Shao J, Wang H, Tao X, Zhu G.
europepmc +1 more source
Derivatives and analogues of benzaldehyde selectively cytotoxic to SV-40 transformed cells.
Jean‐Luc Zundel+2 more
openalex +2 more sources
Suppression of Electroreductive Dimerization of Benzaldehyde by Addition of α-Cyclodextrin [PDF]
Tomokazu Matsue+3 more
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Several derivatives incorporating five‐membered aromatic rings are described in this review as bile acid receptor modulators, particularly targeting the farnesoid X receptor and the G protein‐coupled bile acid receptor 1. This review provides a comprehensive analysis of patents and literature that is useful to support researchers in the design of new ...
Claudia Finamore+5 more
wiley +1 more source
Characterization of Physicochemical Quality and Volatiles in Donkey Meat Hotpot Under Different Boiling Periods. [PDF]
Sun L+9 more
europepmc +1 more source
Continuous Flow Block Copolymer Nanoaggregate Synthesis and Their Flow Dialysis Purification
This work details the methodology for the synthesis of block copolymer nanoparticles through continuous flow self‐assembly and purification via flow dialysis. Nanoaggregates are formed by mixing block copolymer solutions in THF with water, followed by dialysis to eliminate excess solvent.
Gayathri Dev Ammini+2 more
wiley +1 more source
Non-Destructive Determination of Starch Gelatinization, Head Rice Yield, and Aroma Components in Parboiled Rice by Raman and NIR Spectroscopy. [PDF]
Taghinezhad E+8 more
europepmc +1 more source
The Liquid-Phase Oxidation of Benzaldehyde in Benzene
T. Takeuchi, Tetsuo Osa
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Solvent Intensification Effects on the S1(nπ*)←S0Absorption Spectra of Benzaldehyde in Fluid Solutions [PDF]
Kenichi Nakashima, Motohiko Koyanagi
openalex +1 more source