Pegylation approach applied to erlotinib-carbonic anhydrase inhibitors hybrids towards anticancer agents. [PDF]
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Rational Design and Antimycobacterial Evaluation of Aryl Sulfonamide-Linked Isoniazid Hydrazones Against Mycobacterium Tuberculosis. [PDF]
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In-silico studies, synthesis, and pharmacological screening of novel multitarget diphenylpyrazole scaffold as EGFR/BRAF and cyclooxygenase-2 inhibitors. [PDF]
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N-(?5-Cyclopentadienylvanadium)benzenesulfonamide
Russian Chemical Bulletin, 1993N-(η5-Cyclopentadienylvanadium)benzenesulfonamide has been synthesized for the first time by treating benzenesulfonamide orN-(tributylstannyl)benzenesulfonamide with vanadocene.
A S Gordetsov, S V Zimina, S E Skobeleva
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Styrylquinoline derivatives are demonstrated to be HIV-1 integrase inhibitors. On the basis of our previous CoMFA analysis of a series of styrylquinoline derivatives, N-[(2-substituted-styryl)-5-chloro-8-hydroxyquinolin-7-yl]-benzenesulfonamide ...
Cheng-Chu Zeng +2 more
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Synthesis of benzenesulfonamide serinol by the Hinsberg reaction
Ministry of Science and Technology, Vietnam, 2022This research focused on synthesising benzenesulfon-amide serinol (BSSe), a new sulfonamide monomer, by the Hinsberg reaction between primary amine of serinol and sulfonyl of benzenesulfonyl chloride (BSC) in an al-kaline environment. The effect of the reacted environ-ment on the reaction efficiency and structure of BSSe were investigated.
Vu Viet Linh Nguyen +3 more
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Inhibition of β-carbonic anhydrases with ureido-substituted benzenesulfonamides
Bioorganic & Medicinal Chemistry Letters, 2011A series of sulfonamides was prepared by reaction of sulfanilamide with aryl/alkyl isocyanates. The ureido-substituted benzenesulfonamides showed a very interesting profile for the inhibition of several carbonic anhydrases (CAs, EC 4.2.1.1) such as the human hCA II and three β-CAs from pathogenic fungal or bacterial species. The Candida albicans enzyme
F. Pacchiano +4 more
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Benzoxazole benzenesulfonamides as allosteric inhibitors of fructose-1,6-bisphosphatase
Bioorganic & Medicinal Chemistry Letters, 2006AbstractChemInform is a weekly Abstracting Service, delivering concise information at a glance that was extracted from about 200 leading journals. To access a ChemInform Abstract, please click on HTML or PDF.
Chunqiu, Lai +6 more
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Synthesis and Characterization of Benzenesulfonyl Hydrazones and Benzenesulfonamides
Synthetic Communications, 2006Abstract In the search for structural cyclic imide analogues of therapeutic interest, the syntheses and characterization of benzenesulfonyl hydrazones and benzenesulfonamides are described. The benzenesulfonyl chlorides (2) and (3) were obtained through the Diels–Alder reaction between N‐p‐chloro‐sulfonylfenylmaleimide (1) and furan or 2‐methylfuran ...
Kely Navakoski de Oliveira +1 more
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Design and synthesis of C60–benzenesulfonamide conjugates
Tetrahedron Letters, 2010Abstract Synthesis of C 60 –benzenesulfonamide conjugates is reported. The strategies for improving their water solubility, as required for binding to human carbonic anhydrase II, are discussed.
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