Results 171 to 180 of about 8,103 (214)

Pegylation approach applied to erlotinib-carbonic anhydrase inhibitors hybrids towards anticancer agents. [PDF]

open access: yesRSC Med Chem
Filiberti S   +12 more
europepmc   +1 more source

Rational Design and Antimycobacterial Evaluation of Aryl Sulfonamide-Linked Isoniazid Hydrazones Against Mycobacterium Tuberculosis. [PDF]

open access: yesChemMedChem
Kadima MG   +10 more
europepmc   +1 more source

In-silico studies, synthesis, and pharmacological screening of novel multitarget diphenylpyrazole scaffold as EGFR/BRAF and cyclooxygenase-2 inhibitors. [PDF]

open access: yesSci Rep
Abdelgawad MA   +10 more
europepmc   +1 more source

N-(?5-Cyclopentadienylvanadium)benzenesulfonamide

Russian Chemical Bulletin, 1993
N-(η5-Cyclopentadienylvanadium)benzenesulfonamide has been synthesized for the first time by treating benzenesulfonamide orN-(tributylstannyl)benzenesulfonamide with vanadocene.
A S Gordetsov, S V Zimina, S E Skobeleva
exaly   +2 more sources

Design, Synthesis and Anti-HIV Integrase Evaluation of N-(5-Chloro-8-Hydroxy-2-Styrylquinolin-7-yl)Benzenesulfonamide Derivatives

open access: yesMolecules, 2010
Styrylquinoline derivatives are demonstrated to be HIV-1 integrase inhibitors. On the basis of our previous CoMFA analysis of a series of styrylquinoline derivatives, N-[(2-substituted-styryl)-5-chloro-8-hydroxyquinolin-7-yl]-benzenesulfonamide ...
Cheng-Chu Zeng   +2 more
exaly   +3 more sources

Synthesis of benzenesulfonamide serinol by the Hinsberg reaction

Ministry of Science and Technology, Vietnam, 2022
This research focused on synthesising benzenesulfon-amide serinol (BSSe), a new sulfonamide monomer, by the Hinsberg reaction between primary amine of serinol and sulfonyl of benzenesulfonyl chloride (BSC) in an al-kaline environment. The effect of the reacted environ-ment on the reaction efficiency and structure of BSSe were investigated.
Vu Viet Linh Nguyen   +3 more
openaire   +1 more source

Inhibition of β-carbonic anhydrases with ureido-substituted benzenesulfonamides

Bioorganic & Medicinal Chemistry Letters, 2011
A series of sulfonamides was prepared by reaction of sulfanilamide with aryl/alkyl isocyanates. The ureido-substituted benzenesulfonamides showed a very interesting profile for the inhibition of several carbonic anhydrases (CAs, EC 4.2.1.1) such as the human hCA II and three β-CAs from pathogenic fungal or bacterial species. The Candida albicans enzyme
F. Pacchiano   +4 more
openaire   +3 more sources

Benzoxazole benzenesulfonamides as allosteric inhibitors of fructose-1,6-bisphosphatase

Bioorganic & Medicinal Chemistry Letters, 2006
AbstractChemInform is a weekly Abstracting Service, delivering concise information at a glance that was extracted from about 200 leading journals. To access a ChemInform Abstract, please click on HTML or PDF.
Chunqiu, Lai   +6 more
openaire   +2 more sources

Synthesis and Characterization of Benzenesulfonyl Hydrazones and Benzenesulfonamides

Synthetic Communications, 2006
Abstract In the search for structural cyclic imide analogues of therapeutic interest, the syntheses and characterization of benzenesulfonyl hydrazones and benzenesulfonamides are described. The benzenesulfonyl chlorides (2) and (3) were obtained through the Diels–Alder reaction between N‐p‐chloro‐sulfonylfenylmaleimide (1) and furan or 2‐methylfuran ...
Kely Navakoski de Oliveira   +1 more
openaire   +1 more source

Design and synthesis of C60–benzenesulfonamide conjugates

Tetrahedron Letters, 2010
Abstract Synthesis of C 60 –benzenesulfonamide conjugates is reported. The strategies for improving their water solubility, as required for binding to human carbonic anhydrase II, are discussed.
Tatiana Y. Zakharian   +1 more
openaire   +1 more source

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