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Benzenesulfonamide analogs of fluoroquinolones. Antibacterial activity and QSAR studies
European Journal of Medicinal Chemistry, 2005The structure-activity relationships (SAR) of new antibacterial benzenesulfonamidefluoroquinolones (BSFQs), coming from derivatization of N4-piperazinyl of ciprofloxacin (CIP) were studied. The behavior of the new BSFQ series was similar to the previously norfloxacin (NOR) analogs reported, making possible a quantitative structure-activity ...
M J, Nieto +3 more
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2012
[6536-23-8] C6H5NO3S2 (MW 203.24) InChI = 1S/C6H5NO3S2/c8-11-7-12(9,10)6-4-2-1-3-5-6/h1-5H InChIKey = BTUNHNFBTGHBRC-UHFFFAOYSA-N (reagent used in a wide array of ene-reactions and cycloadditions) Physical Data: mp 73 °C; bp 110–120 °C at 0.004 mbar.
Philipp Heretsch, Athanassios Giannis
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[6536-23-8] C6H5NO3S2 (MW 203.24) InChI = 1S/C6H5NO3S2/c8-11-7-12(9,10)6-4-2-1-3-5-6/h1-5H InChIKey = BTUNHNFBTGHBRC-UHFFFAOYSA-N (reagent used in a wide array of ene-reactions and cycloadditions) Physical Data: mp 73 °C; bp 110–120 °C at 0.004 mbar.
Philipp Heretsch, Athanassios Giannis
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Metal-Free Amidation Reactions of Terminal Alkynes with Benzenesulfonamide
The Journal of Organic Chemistry, 2019A novel and efficient approach has been developed to synthesize α-sulfonylamino ketones through the reaction between terminal alkynes and sulfonamides under ambient air using PIDA (diacetoxy iodobenzene). A library of α-sulfonylamino ketone derivatives having a variety of substituents has been synthesized.
Sachinta Mahato +3 more
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NMR studies of carbonic anhydrase-fluorinated benzenesulfonamide complexes
Biochemistry, 1989Fluorine NMR has been used to examine complexes formed by 2-fluoro-, 3-fluoro-, and 2,5-difluorobenzenesulfonamide and human carbonic anhydrases I and II. The results show that all three inhibitors form complexes with both isozymes that have 2:1 inhibitor/enzyme stoichiometry.
L B, Dugad, C R, Cooley, J T, Gerig
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Antiparkinsonian activity of benzenesulfonamide derivatives — selective MAO-B inhibitors
Bulletin of Experimental Biology and MedicineThe anti-parkinsonian activity of benzolsulfonamide selective MAO-B inhibitors was evaluated in a model of experimental parkinsonism in white mice (systemic administration of 1-methyl-4-phenyl-1,2,3,6-tetrahydropyridine; MPTP). Six candidate compounds (laboratory codes S6-S8 and S11-S13) were analyzed. Rasagiline was used as the reference drug.
A L, Khokhlov +7 more
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N-Heterocyclic Benzenesulfonamides
Journal of the American Chemical Society, 1951Martin E. Hultquist +6 more
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