Results 261 to 270 of about 767,969 (287)

The BET inhibitor JQ1 attenuates double-strand break repair and sensitizes models of pancreatic ductal adenocarcinoma to PARP inhibitors

EBioMedicine, 2019
Patrick L Garcia, Robert C A M van Waardenburg, Karina Yoon   +2 more
exaly  

Synergistic activity of BET inhibitor BI 894999 with PLK inhibitor volasertib in AML and

Cancer Letters, 2018
Harald Engelhardt, Daniel Gerlach, Norbert Kraut   +2 more
exaly  

Structure-guided discovery of a novel, potent, and orally bioavailable 3,5-dimethylisoxazole aryl-benzimidazole BET bromodomain inhibitor

Bioorganic and Medicinal Chemistry, 2019
Richard L Mackman, Jeff Zablocki, Anita Niedziela-Majka   +2 more
exaly  

Harnessing BET Inhibitor Sensitivity Reveals AMIGO2 as a Melanoma Survival Gene

Molecular Cell, 2017
Pamela Wu, Dan Filipescu, Emily Bernstein   +2 more
exaly  

The BET bromodomain inhibitor JQ1 radiosensitizes non-small cell lung cancer cells by upregulating p21

Cancer Letters, 2017
Gang Wu, Jian Wang, Hong Mei
exaly  

CRYSTALLINE SOLID FORMS OF A BET INHIBITOR

2017
CHEN SHILI, JIA ZHONGJIANG, LIU PINGLI, QIAO LEI, WU YONGZHONG, ZHOU JIACHENG, LI QUN   +6 more
openaire   +7 more sources

TRICYCLIC HETEROCYCLES AS BET PROTEIN INHIBITORS

2014
COMBS ANDREW P, SPARKS RICHARD B, MADUSKUIE JR THOMAS P, RODGERS JAMES D   +3 more
openaire   +10 more sources

Assessment of the Antiproliferative Activity of a BET Bromodomain Inhibitor as Single Agent and in Combination in Non-Hodgkin Lymphoma Cell Lines

Methods in Molecular Biology, 2016
Francesco Bertoni, Eugenio Gaudio, Ivo Kwee   +2 more
exaly  

Targeting AMPK-ULK1-mediated autophagy for combating BET inhibitor resistance in acute myeloid leukemia stem cells

Autophagy, 2017
Jung Yeon Lee, Yoo Hong Min, Jieun Jang
exaly  

A new BET inhibitor, 171, inhibits tumor growth through cell proliferation inhibition more than apoptosis induction

Investigational New Drugs, 2019
Mohammadali Soleimani Damaneh, Bing Xiong, Tao Meng   +2 more
exaly