Results 191 to 200 of about 27,094 (219)

Overexpression of bromodomain factor 3 in Trypanosoma cruzi (TcBDF3) affects differentiation of the parasite and protects it against bromodomain inhibitors

FEBS Journal, 2016
Pamela Cribb, Victoria Lucia Alonso, Julia A Cricco   +2 more
exaly  

BROMODOMAIN INHIBITORS

2013
WANG LE, PRATT JOHN K, MCDANIEL KEITH F, DAI YUJIA, FIDANZE STEVEN D, HASVOLD LISA, HOLMS JAMES H, KATI WARREN M, LIU DACHUN, MANTEI ROBERT A, MCCLELLAN WILLIAM J, SHEPPARD GEORGE S, WADA CAROL K   +12 more
openaire   +7 more sources

Bromodomain inhibitors, JQ1 and I-BET 762, as potential therapies for pancreatic cancer

Cancer Letters, 2017
Ana Sofia Mendes Leal, Patricia A Pioli, Karen T Liby   +2 more
exaly  

A Series of Potent CREBBP Bromodomain Ligands Reveals an Induced-Fit Pocket Stabilized by a Cation–π Interaction†

Angewandte Chemie - International Edition, 2014
Oleg L. Fedorov, Stefan Knapp, Timothy Rooney   +2 more
exaly  

Bromodomain

2008
openaire   +2 more sources

The structural basis for the recognition of acetylated histone H4 by the bromodomain of histone acetyltransferase Gcn5p

EMBO Journal, 2000
Patrizia Filetici, David J. Owen, David Neuhaus   +2 more
exaly  

BET bromodomain inhibitors: a patent review

Expert Opinion on Therapeutic Patents, 2014
Christopher J. Burns, Phillip P. Sharp
exaly  

1,3-Dimethyl Benzimidazolones Are Potent, Selective Inhibitors of the BRPF1 Bromodomain

ACS Medicinal Chemistry Letters, 2014
Paul Bamborough, Chun-Wa Chung, Rab K Prinjha   +2 more
exaly  

Discovery of alkoxy benzamide derivatives as novel BPTF bromodomain inhibitors via structure-based virtual screening

Bioorganic Chemistry, 2019
Chun-Shen Zhao, Wenchao Lu, Cheng Luo
exaly  

Androgen Receptor Deregulation Drives Bromodomain-Mediated Chromatin Alterations in Prostate Cancer

Cell Reports, 2017
Ian G Mills, Stefan Knapp, Matti Nykter
exaly