Results 221 to 230 of about 33,428 (239)

LP99: Discovery and Synthesis of the First Selective BRD7/9 Bromodomain Inhibitor

Angewandte Chemie - International Edition, 2015
Lucas C C Vieira, Cynthia Tallant, Oleg Fedorov   +2 more
exaly  

Overexpression of bromodomain factor 3 in Trypanosoma cruzi (TcBDF3) affects differentiation of the parasite and protects it against bromodomain inhibitors

FEBS Journal, 2016
Victoria Lucia Alonso, Pamela Cribb, Julia A Cricco   +2 more
exaly  

A Series of Potent CREBBP Bromodomain Ligands Reveals an Induced‐Fit Pocket Stabilized by a Cation–π Interaction

Angewandte Chemie - International Edition, 2014
Timothy P C Rooney, Panagis Filippakopoulos, Oleg Fedorov   +2 more
exaly  

Bromodomain inhibitors, JQ1 and I-BET 762, as potential therapies for pancreatic cancer

Cancer Letters, 2017
Ana S Leal, Charlotte R Williams, Darlene B Royce   +2 more
exaly  

The structural basis for the recognition of acetylated histone H4 by the bromodomain of histone acetyltransferase Gcn5p

EMBO Journal, 2000
P R Evans, David Neuhaus, Patrizia Filetici   +2 more
exaly  

BET bromodomain inhibitors: a patent review

Expert Opinion on Therapeutic Patents, 2014
Jean-Marc Garnier, Phillip P Sharp, Christopher J Burns   +2 more
exaly  

1,3-Dimethyl Benzimidazolones Are Potent, Selective Inhibitors of the BRPF1 Bromodomain

ACS Medicinal Chemistry Letters, 2014
Paul Bamborough, Chun-Wa Chung, Peter D Craggs   +2 more
exaly  

The transcriptional regulation role of BRD7 by binding to acetylated histone through bromodomain

Journal of Cellular Biochemistry, 2006
Xiao Ling Li
exaly  

Bromodomain

2006
openaire   +1 more source

Discovery of alkoxy benzamide derivatives as novel BPTF bromodomain inhibitors via structure-based virtual screening

Bioorganic Chemistry, 2019
Dan Zhang, Wenchao Lu, Fulin Lian
exaly