Results 121 to 130 of about 632,694 (239)

Deep Learning Dynamic Allostery of G‑Protein-Coupled Receptors

JACS Au, 2023
Hung N. Do, Jinan Wang, Yinglong Miao
doaj   +1 more source

Domains involved in the specificity of G protein activation in phospholipase C-coupled metabotropic glutamate receptors.

, 1994
Jean‐Philippe Pin, C. Joly, Stephen F. Heinemann, Joël Bockaert   +3 more
openalex   +1 more source

Inclusion of Enclosed Hydration Effects in the Binding Free Energy Estimation of Dopamine D3 Receptor Complexes

, 2019
Confined hydration and conformational flexibility are some of the challenges encountered for the rational design of selective antagonists of G-protein coupled receptors. We present a set of C3-substituted (-)-stepholidine derivatives as potent binders of
Cordone, Pierpaolo, Gadhiya, Satishkumar, Gallicchio, Emilio, Harding, Wayne W., Kurtzman, Tom, Pal, Rajat Kumar, Ramsey, Steve, Wickstrom, Lauren   +7 more
core   +2 more sources

A Truncated Form of RGS3 Negatively Regulates G Protein-coupled Receptor Stimulation of Adenylyl Cyclase and Phosphoinositide Phospholipase C [PDF]

, 1997
Tapan K. Chatterjee, Alex Eapen, Rory A. Fisher   +2 more
openalex   +1 more source

A human gene encodes a putative G protein-coupled receptor highly expressed in the central nervous system [PDF]

, 1998
Patrick J. Donohue, Hagit Shapira, Samuel A. Mantey, Lori L. Hampton, Robert T. Jensen, James F. Battey   +5 more
openalex   +1 more source

Thyrotropin-releasing hormone activates Ca2+ efflux. Evidence suggesting that a plasma membrane Ca2+ pump is an effector for a G-protein-coupled Ca(2+)-mobilizing receptor.

, 1994
Eric J. Nelson, Patricia M. Hinkle
openalex   +1 more source

Reciprocal In Vivo Regulation of Myocardial G Protein–Coupled Receptor Kinase Expression by β-Adrenergic Receptor Stimulation and Blockade [PDF]

, 1998
Guido Iaccarino, Eric D. Tomhave, Robert J. Lefkowitz, Walter J. Koch   +3 more
openalex   +1 more source

Potential Regulatory Roles for G Protein-Coupled Receptor Kinases and -Arrestins in Gonadotropin-Releasing Hormone Receptor Signaling [PDF]

, 1998
Jimmy D. Neill
openalex   +1 more source

Inhibition of thrombin receptor signaling by a G-protein coupled receptor kinase. Functional specificity among G-protein coupled receptor kinases.

, 1994
Kenji Ishii, J. Chen, Maki Ishii, Walter J. Koch, Neil J. Freedman, R J Lefkowitz, Shaun R. Coughlin   +6 more
openalex   +1 more source

Identification by polymerase chain reaction of the G protein-coupled receptor kinases expressed in the mouse gonadotropic alpha T3-1 cell line. [PDF]

, 1996
Jimmy D. Neill, Lois C. Musgrove, Jeffrey C. Sellers, L. Wayne Duck   +3 more
openalex   +1 more source