Results 101 to 110 of about 3,102 (198)

Novel naphthyridines are histamine H3 antagonists and serotonin reuptake transporter inhibitors

, 2007
Michael A. Letavic, John M. Keith, Kiev S. Ly, Ann Barbier, Jamin D. Boggs, Sandy J. Wilson, Brian Lord, Timothy W. Lovenberg, Nicholas I. Carruthers   +8 more
openalex   +1 more source

In vitro SAR of pyrrolidine-containing histamine H3 receptor antagonists: Trends across multiple chemical series

, 2007
Diana L. Nersesian, Lawrence A. Black, Thomas R. Miller, Timothy A. Vortherms, Timothy A. Esbenshade, Arthur A. Hancock, Marlon Cowart   +6 more
openalex   +1 more source

Synthesis and structure–activity relationships of 4,5-fused pyridazinones as histamine H3 receptor antagonists

, 2011
Ming Tao, Rita Raddatz, Lisa D. Aimone, Robert L. Hudkins   +3 more
openalex   +1 more source

In vitro studies on a class of quinoline containing histamine H3 antagonists

, 2010
Huaqing Liu, Robert J. Altenbach, Gilbert Diaz, Arlene M. Manelli, Ruth L. Martin, Thomas R. Miller, Timothy A. Esbenshade, Jorge D. Brioni, Marlon Cowart   +8 more
openalex   +1 more source

Development and Preclinical Characterization of [¹⁸F]H3-2406 and [¹⁸F]H3-2407 for Positron Emission Tomography Imaging of the Histamine Subtype-3 Receptor. [PDF]

J Med Chem
Song Z, Li Y, Dahl K, Sun Z, Chen J, Zhou X, Gao Y, Rong J, Zhao C, Yuan K, Chaudhary AF, Patel JS, Collier TL, Ran C, Muehlfenzl KS, Haider A, Elmore CS, Schou M, Liang SH.   +18 more
europepmc   +1 more source

A new class of histamine H3 receptor antagonists derived from ligand based design

, 2007
Olivier Roche, Rosa Marı́a Rodrı́guez Sarmiento   +1 more
openalex   +1 more source

Improvement of the Prediction Power of the CoMFA and CoMSIA Models on Histamine H3 Antagonists by Different Variable Selection Methods. [PDF]

Sci Pharm, 2012
Ghasemi JB, Tavakoli H.
europepmc   +1 more source

0624 Anticataplectic Efficacy of Pitolisant, the First Potent and Highly Selective Histamine H3-Receptor Antagonist/Inverse Agonist [PDF]

, 2018
Michael J. Thorpy, J. Schwartz, J Lecomte, Sébastien Causse, Jeffrey M. Dayno   +4 more
openalex   +1 more source

Subtype-specific dysregulation of biogenic amine-related genes and miRNAs in breast cancer: identification of DRD2, HRH2, and HRH4 as potential therapeutic targets in TNBC and HER2+ subtypes. [PDF]

Breast Cancer Res Treat
Sirek A, Sirek T, Nowakowski R, Borawski P, Ossowski P, Mitka-Krysiak E, Zmarzły N, Boroń K, Chalcarz M, Kuraszewska B, Szulik M, Boroń D, Grabarek BO.   +12 more
europepmc   +1 more source

A Radiolabeled Photoswitchable G Protein-Coupled Receptor Antagonist Enlightens Ligand Binding Kinetics Associated with Photoswitching. [PDF]

J Am Chem Soc
Binkhorst LCP, Josimovic I, De Boer B, Simon IA, Van Der Aa F, Zarzycka BA, De Esch IJP, Vischer HF, Windhorst AD, Wijtmans M, Leurs R.   +10 more
europepmc   +1 more source