Results 121 to 130 of about 3,102 (198)

Discovery of novel steroidal histamine H3 receptor antagonists/inverse agonists. Part 2. Versatile steroidal carboxamide derivatives

, 2019
István Ledneczki, Zsolt Némethy, Pál Tapolcsányi, János Éles, István Greiner, Eszter Gábor, Balázs Varga, Ottilia Balázs, Viktor Román, György Lévay, Sándor Mahó   +10 more
openalex   +1 more source

The Histamine-Associated Inflammatory Landscape of Endometriosis: Molecular Profiling of HDC, HRH1-HRH4, and Cytokines Across Lesion Subtypes. [PDF]

Int J Mol Sci
Velho RV, Freitag JH, Brueckner AM, Thalmeier L, Pohl J, Mechsner S.   +5 more
europepmc   +1 more source

Influence of the antagonists LINS01005 and LINS01007 on histamine H3 / H4 receptors in murine asthma model

, 2019
Leandro Kanamaru Franco de [UNESP] Lima
openalex   +1 more source

Characterisation of the specific binding of the histamine H3 receptor antagonist radioligand [3H]GR168320

, 1996
Jason Brown, Celestine T. O’Shaughnessy, Gavin J. Kilpatrick, D. I. C. SCOPES, Paul Beswick, John W. Clitherow, Julie C. Barnes   +6 more
openalex   +1 more source

Emerging Epigenetic Therapeutics and Diagnostics for Autism Spectrum Disorder. [PDF]

Curr Issues Mol Biol
Kao C, Lim KK, Chen ES.
europepmc   +1 more source

Virtual Screening Approaches to Identify Promising Multitarget-Directed Ligands for the Treatment of Autism Spectrum Disorder. [PDF]

Molecules
Jończyk J, Przybylska K, Staszewski M, Godyń J, Werner T, Stefaniak-Napieralska M, Stark H, Walczyński K, Bajda M.   +8 more
europepmc   +1 more source

Pre-clinical characterization of aryloxypyridine amides as histamine H3 receptor antagonists: Identification of candidates for clinical development

, 2010
Michael A. Letavic, Leah Aluisio, John Atack, Pascal Bonaventure, Nicholas I. Carruthers, Christine Dugovic, Anita Everson, Mark A. Feinstein, Ian Fraser, Kenway Hoey, Xiaohui Jiang, John M. Keith, Tatiana Koudriakova, Perry Leung, Brian Lord, Timothy W. Lovenberg, Kiev S. Ly, Kirsten L. Morton, S. Timothy Motley, Diane Nepomuceno, Michèle Rizzolio, Raymond Rynberg, Kia Sepassi, Jonathan Shelton   +23 more
openalex   +1 more source

Screening and identification of the H1R antagonists from natural products by BODIPY FL histamine recognition and DPHD-anchored bombardment coupled with target cell extraction. [PDF]

Front Pharmacol
Li X, Hu G, Chen X, Di C, Qi J.
europepmc   +1 more source

Pharmacological characterization of GT-2016, a non-thiourea-containing histamine H3 receptor antagonist: in vitro and in vivo studies.

, 1995
Clark E. Tedford, Stephen L. Yates, G Pawłowski, Julia W. Nalwalk, Lindsay B. Hough, M. Khan, James G. Phillips, G. J. DURANT, Robert C.A. Frederickson   +8 more
openalex   +1 more source

Molecular Insights into Bromocriptine Binding to GPCRs Within Histamine-Linked Signaling Networks: Network Pharmacology, Pharmacophore Modeling, and Molecular Dynamics Simulation. [PDF]

Int J Mol Sci
Dermawan D, Elbouamri L, Chtita S, Alotaiq N.   +3 more
europepmc   +1 more source