Anti-proliferate Activity and 5α-reductase Inhibitors of Chiral Macrocyclic (Nα-di-nicotinoyl)[L-phenylalaninyl-L-leucinyl]Pentapeptide Candidates Against LNCaP and PC-3 Prostate Cancer Cell Lines [PDF]
60-65A series of macrocyclic derivatives 2-6 were prepared using Nα-dinicotinoyl-bis[L-phenylalaninyl-L-leucyl]hydrazide 1 and cyclo pentapeptide hydrazide 2 as starting materials.
Alanazi, M M+4 more
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In the present study, a rapid, less expensive, clean and environmental friendly route to synthesis new pyrazoles, pyrazolopyridazines and condensed pyrimidines was developed via grinding of 2-(3-(dimethylamino)acryloyl)-3H-benzo[f]chromen-3-one (1) with ...
Anhar Abdel-Aziem+3 more
doaj +1 more source
Bio-Based (Chitosan-ZnO) Nanocomposite: Synthesis, Characterization, and Its Use as Recyclable, Ecofriendly Biocatalyst for Synthesis of Thiazoles Tethered Azo Groups. [PDF]
Bashal AH+5 more
europepmc +1 more source
(3+2)-Cycloadditions of Levoglucosenone (LGO) with Fluorinated Nitrile Imines Derived from Trifluoroacetonitrile: An Experimental and Computational Study. [PDF]
Mlostoń G+4 more
europepmc +1 more source
Regioselective Cycloaddition of Nitrile Imines to 5-Methylidene-3-phenyl-hydantoin: Synthesis and DFT Calculations. [PDF]
Filkina ME+5 more
europepmc +1 more source
Preparation of 1,3,5-Trisubstituted Pyrazoles with Cascade Reaction Catalyzed by Cu between Hydrazonoyl Halide and Terminal Alkynes [PDF]
Fuwei Li, Xiaolong Wang, Haitao Yu
openalex +1 more source
p-Aminobenzoic acid chitosan/CuONPs (ACs/CuONPs) composites, developed using chitosan (Cs) and its grafted form (ACs), proved to be efficient, eco-friendly catalysts for synthesizing novel bisthiazole and bisthiadiazole derivatives.
Mohamed El-Naggar+7 more
doaj +1 more source
One-Pot Synthesis of 1-Aryl-3-trifluoromethylpyrazoles Using Nitrile Imines and Mercaptoacetaldehyde As a Surrogate of Acetylene. [PDF]
Świątek K+4 more
europepmc +1 more source
Synthesis, Charactrization and Evaluation Biological Activity of some New Formazan Compounds Derived from Schiff Bases and Azo Compounds [PDF]
The titled compounds (( twenty compounds )) were synthesized from series reactions of two types compounds ( azo and imine ) - compounds ., we prepared ten compounds from Schiff bases which react after that with diazo ...
Abad Shallal, Mohammed+1 more
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Computational studies on formation and intermolecular [1+2] cycloadditions of nitrilimines [PDF]
2,5-disubstituted tetrazoles decompose thermally to give nitrilimines (R1–CNN–R2), whose electronic structure widely varies with the substituents R1 and R2.
Mehrpajouh, Sima
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