Results 1 to 10 of about 15,973 (252)

Reactions of acryl thioamides with iminoiodinanes as a one-step synthesis of <i>N</i>-sulfonyl-2,3-dihydro-1,2-thiazoles. [PDF]

Beilstein J Org Chem
A one-step method has been developed for the preparation of 2,3-dihydro-2-sulfonyl-3,4,5-substituted 1,2-thiazoles by the reaction of acryl thioamides and iminoiodinanes.
Ilkin VG, Silaichev PS, Filimonov VO, Beryozkina TV, Likhacheva MD, Slepukhin PA, Dehaen W, Bakulev VA.   +7 more
europepmc   +2 more sources

Thiazolylcyanocyclopropanes: Novel Donor-Acceptor Cyclopropanes for Accessing Thiazole-Containing Targets. [PDF]

Molecules
Donor–acceptor (D–A) cyclopropanes are important precursors in the synthesis of complex molecules due to their bidentate character and high reactivity.
Savini EB, Bandieri E, Pecchini P, Santarelli N, Bernardi L, Fochi M.   +5 more
europepmc   +2 more sources

Novel hybrid thiazoles, bis-thiazoles linked to azo-sulfamethoxazole: Synthesis, docking, and antimicrobial activity

Heliyon
The reaction of sulfamethoxazolehydrazonoyl chloride with thiosemicarbazones, bis-thiosemicarbazones, or 4-amino-3-mercapto-1,2,4-triazole in dioxane in the presence of triethylamine as a basic catalyst at reflux resulted in the regioselective synthesis ...
Faisal K Algethami, Mohamed Attia Ragheb, Ahmed H M Elwahy   +2 more
exaly   +3 more sources

3-Phenylpropanal and citral in the multicomponent synthesis of novel thiopyrano[2,3-d]thiazoles

Results in Chemistry, 2022
A 3-phenylpropanal and citral were studied in the multicomponent reaction with the isorhodanine and maleimides (EDDA catalyst) with the aim of the novel thiopyrano[2,3-d]thiazoles synthesis.
Andrii Lozynskyi, Andriy Karkhut, Svyatoslav Polovkovych, Olexandr Karpenko, Serhii Holota, Andrzej K. Gzella, Roman Lesyk   +6 more
doaj   +1 more source

Pyridin-2-ylthiazolothiazoles – Synthesis and photophysical properties

Results in Chemistry, 2021
Thiazolo[5,4-d]thiazoles are valuable materials for a range of technical and biological applications. They are used as chemosensors, electroluminescent materials, organic light-emitting diodes (OLEDs), in solar cells, in live-cell imaging, etc., and for ...
Ana F.R. Cerqueira, Maria G.P.M.S. Neves, A. Jorge Parola, Augusto C. Tomé   +3 more
doaj   +1 more source

Thiazole Ring—A Biologically Active Scaffold

Molecules, 2021
Background: Thiazole is a good pharmacophore nucleus due to its various pharmaceutical applications. Its derivatives have a wide range of biological activities such as antioxidant, analgesic, and antimicrobial including antibacterial, antifungal ...
Anthi Petrou, Maria Fesatidou, Athina Geronikaki   +2 more
doaj   +1 more source

Synthesis of Novel Thiazole Derivatives Bearing β-Amino Acid and Aromatic Moieties as Promising Scaffolds for the Development of New Antibacterial and Antifungal Candidates Targeting Multidrug-Resistant Pathogens

Molecules, 2021
Rapidly growing antimicrobial resistance among clinically important bacterial and fungal pathogens accounts for high morbidity and mortality worldwide.
Dovilė Malūkaitė, Birutė Grybaitė, Rita Vaickelionienė, Giedrius Vaickelionis, Birutė Sapijanskaitė-Banevič, Povilas Kavaliauskas, Vytautas Mickevičius   +6 more
doaj   +1 more source

Photochemical permutation of thiazoles, isothiazoles and other azoles. [PDF]

Nature
Roure B, Alonso M, Lonardi G, Yildiz DB, Buettner CS, Dos Santos T, Xu Y, Bossart M, Derdau V, Méndez M, Llaveria J, Ruffoni A, Leonori D.   +12 more
europepmc   +2 more sources

Novel Structural Hybrids of Pyrrole and Thiazole Moieties: Synthesis and Evaluation of Antibacterial and Antifungal Activities

Acta Chimica Slovenica, 2021
One of the best ways to design new biocidal agents is synthesizing hybrid molecules by combining two or more bioactive moieties in a single molecular scaffold.
Mohamed Salem, Samir Abbas, Marwa El-Sharief, Mohamed Helal, Moustafa Gouda, Mohammed Assiri, Mohammed Assiri, Tarik Ali, Tarik Ali   +8 more
doaj   +1 more source

Ultrasound-assisted green synthesis and antimicrobial assessment of 1,3-thiazoles and 1,3,4-thiadiazines

Green Chemistry Letters and Reviews, 2021
In this article, we applied ultrasonic irradiation as an ecofriendly, green, efficient approach for the synthesis of a new 1,3-thiazoles and 1,3,4-thiadiazines under solvent-free conditions.
Sara N. Shabaan, Basma Saad Baaiu, Anhar Abdel-Aziem, Mohamed S. Abdel-Aziz   +3 more
doaj   +1 more source