Results 1 to 10 of about 9,832 (211)

Reactions of acryl thioamides with iminoiodinanes as a one-step synthesis of N-sulfonyl-2,3-dihydro-1,2-thiazoles [PDF]

Beilstein Journal of Organic Chemistry
A one-step method has been developed for the preparation of 2,3-dihydro-2-sulfonyl-3,4,5-substituted 1,2-thiazoles by the reaction of acryl thioamides and iminoiodinanes.
Vladimir G. Ilkin, Pavel S. Silaichev, Valeriy O. Filimonov, Tetyana V. Beryozkina, Margarita D. Likhacheva, Pavel A. Slepukhin, Wim Dehaen, Vasiliy A. Bakulev   +7 more
doaj   +2 more sources

Thiazolylcyanocyclopropanes: Novel Donor–Acceptor Cyclopropanes for Accessing Thiazole-Containing Targets [PDF]

Molecules
Donor–acceptor (D–A) cyclopropanes are important precursors in the synthesis of complex molecules due to their bidentate character and high reactivity.
Emanuèl Bruno Savini, Edoardo Bandieri, Pietro Pecchini, Nicolò Santarelli, Luca Bernardi, Mariafrancesca Fochi   +5 more
doaj   +2 more sources

Novel hybrid thiazoles, bis-thiazoles linked to azo-sulfamethoxazole: Synthesis, docking, and antimicrobial activity

Heliyon
The reaction of sulfamethoxazolehydrazonoyl chloride with thiosemicarbazones, bis-thiosemicarbazones, or 4-amino-3-mercapto-1,2,4-triazole in dioxane in the presence of triethylamine as a basic catalyst at reflux resulted in the regioselective synthesis ...
Ahmed Elwahy, Magdi E A Zaki, Ismail Abdelshafy Abdelhamid   +2 more
exaly   +3 more sources

3-Phenylpropanal and citral in the multicomponent synthesis of novel thiopyrano[2,3-d]thiazoles

Results in Chemistry, 2022
A 3-phenylpropanal and citral were studied in the multicomponent reaction with the isorhodanine and maleimides (EDDA catalyst) with the aim of the novel thiopyrano[2,3-d]thiazoles synthesis.
Andrii Lozynskyi, Andriy Karkhut, Svyatoslav Polovkovych, Olexandr Karpenko, Serhii Holota, Andrzej K. Gzella, Roman Lesyk   +6 more
doaj   +1 more source

Pyridin-2-ylthiazolothiazoles – Synthesis and photophysical properties

Results in Chemistry, 2021
Thiazolo[5,4-d]thiazoles are valuable materials for a range of technical and biological applications. They are used as chemosensors, electroluminescent materials, organic light-emitting diodes (OLEDs), in solar cells, in live-cell imaging, etc., and for ...
Ana F.R. Cerqueira, Maria G.P.M.S. Neves, A. Jorge Parola, Augusto C. Tomé   +3 more
doaj   +1 more source

Selected 5-amino-1-aryl-1H-1,2,3-triazole scaffolds as promising antiproliferative agents [PDF]

The Ukrainian Biochemical Journal, 2020
Development of a new effective drugs with low side effects and definite chemical characteristics needs indentification of bioactive scaffolds for further structural optimization.
N. Pokhodylo, O. Shyyka, N. Finiuk, R. Stoika   +3 more
doaj   +1 more source

The Synthesis of Novel 2-Hetarylthiazoles via the Stille Reaction

Журнал органічної та фармацевтичної хімії, 2023
A preparative approach to the synthesis of 2-hetaryl thiazoles has been developed via the interaction of halothiazoles with stannanes according to the Stille reaction. The most effective catalysts and reaction conditions have been found.
Dmytro O. Tarasenko, Volodymyr M. Kotliar   +1 more
doaj   +1 more source

5-(4-Methoxyphenyl)-1-[4-(4-methoxyphenyl)thiazol-2-yl]-3-[4-(prop-2-ynyloxy)phenyl]-4,5-dihydro-1H-pyrazole

IUCrData, 2022
The title compound, C29H25N3O3S, crystallizes in the monoclinic space group P21/n. The molecule contains a central four-ring system in which all of the rings are almost coplanar.
Sreeramapura D. Archana, Holalagudu A. Nagma Banu, Balakrishna Kalluraya, Hemmige S. Yathirajan, Rishik Balerao, Ray J. Butcher   +5 more
doaj   +1 more source

The Structure of Biologically Active Functionalized Azoles: NMR Spectroscopy and Quantum Chemistry

Magnetochemistry, 2022
This review summarizes the data on the stereochemical structure of functionalized azoles (pyrazoles, imidazoles, triazoles, thiazoles, and benzazoles) and related compounds obtained by multipulse and multinuclear 1H, 13C, 15N NMR spectroscopy and quantum
Lyudmila I. Larina
doaj   +1 more source

Development of Novel Pyridine-Thiazole Hybrid Molecules as Potential Anticancer Agents

Molecules, 2022
Novel pyridine-thiazole hybrid molecules were synthesized and subjected to physico-chemical characterization and screening of their cytotoxic action towards a panel of cell lines derived from different types of tumors (carcinomas of colon, breast, and ...
Iryna Ivasechko, Ihor Yushyn, Piotr Roszczenko, Julia Senkiv, Nataliya Finiuk, Danylo Lesyk, Serhii Holota, Robert Czarnomysy, Olga Klyuchivska, Dmytro Khyluk, Nataliya Kashchak, Andrzej Gzella, Krzysztof Bielawski, Anna Bielawska, Rostyslav Stoika, Roman Lesyk   +15 more
doaj   +1 more source